Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Thromboxane A2 receptor (MOUSE) | BDBM50353639 (CHEMBL1829806) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353632 (CHEMBL1829812) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353635 (CHEMBL1829801) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353643 (CHEMBL1829808) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353645 (CHEMBL1829810) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353640 (CHEMBL65121) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353638 (CHEMBL1829805) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353636 (CHEMBL1829802) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353646 (CHEMBL1829811) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 259 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353644 (CHEMBL1829809) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 463 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353641 (CHEMBL1829804) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353634 (CHEMBL1828642) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353642 (CHEMBL1829807) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353633 (CHEMBL1829813) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane A2 receptor (MOUSE) | BDBM50353637 (CHEMBL1829803) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pennsylvania Curated by ChEMBL | Assay Description Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono... | J Med Chem 54: 6969-83 (2011) Article DOI: 10.1021/jm200980u BindingDB Entry DOI: 10.7270/Q2H995KG | |||||||||||
More data for this Ligand-Target Pair |