Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197347 (Ebselen Diselenide) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197302 (CHEMBL3920474) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197323 (CHEMBL3931605) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 920 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197313 (CHEMBL3930560) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197299 (CHEMBL3913676) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197303 (CHEMBL3892953) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM34233 (2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197304 (CHEMBL3913688) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197344 (CHEMBL3903564) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197297 (CHEMBL3928799 | ebselen derivative 2d) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197342 (CHEMBL3912637) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197300 (CHEMBL3912164 | ebselen derivative 2e) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197346 (CHEMBL3919905) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197298 (CHEMBL3947694) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197343 (CHEMBL3940582) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197301 (CHEMBL3922662 | ebselen derivative 1d) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.02E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM106945 (US8592468, EbSe3) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197296 (CHEMBL3894673) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.43E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50197345 (CHEMBL3931557) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.19E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Technology Curated by ChEMBL | Assay Description Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ... | Bioorg Med Chem Lett 26: 5254-5259 (2016) Article DOI: 10.1016/j.bmcl.2016.09.050 BindingDB Entry DOI: 10.7270/Q28917T7 | |||||||||||
More data for this Ligand-Target Pair |