Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50014917 (4-(2-Chloro-phenyl)-2-imidazol-1-ylmethyl-6-methyl...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50368043 (CHEMBL1203671) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50368033 (CHEMBL1203626) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50368037 (CHEMBL1744226) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM7962 (4-(2-Imidazol-1-yl-ethoxy)-benzoic acid; hydrochlo...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50368032 (CHEMBL1203662) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50368039 (CHEMBL1202293) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.95E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50014902 (4-(2-Difluoromethoxy-phenyl)-2-imidazol-1-ylmethyl...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50014915 (4-(2-Chloro-3-trifluoromethyl-phenyl)-2-imidazol-1...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thromboxane-A synthase (Homo sapiens (Human)) | BDBM50318494 (3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research UK Curated by ChEMBL | Assay Description Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kg | J Med Chem 33: 646-52 (1990) BindingDB Entry DOI: 10.7270/Q25X29HP | |||||||||||
More data for this Ligand-Target Pair |