Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aromatase (Homo sapiens (Human)) | BDBM8889 (3-(3,4-Dihydronaphthalen-2-yl)pyridine | Dihydrona...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 4.07 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8611 (4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 29.5 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8611 (4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 30 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8611 (4-{5H,6H,7H,8H-imidazo[1,5-a]pyridin-5-yl}benzonit...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 30 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8917 (1-(3-methoxynaphthalen-2-yl)-1H-imidazole | Imidaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 129 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8905 (3-(6-Methoxy-2-naphthyl)pyridine | 3-(6-methoxynap...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 586 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8891 (3-(6-Methoxy-3,4-dihydronaphthalen-2-yl)pyridine |...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 814 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8912 (3-(1,5-Dichloro-6-methoxy-2-naphthyl)pyridine | 3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 970 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8914 (Methyl 6-pyridin-3-yl-2-naphthoate | Pyridine-subs...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents | US Patent | n/a | n/a | 1.25E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8893 (3-(1-Ethyl-3,4-dihydronaphthalen-2-yl)-pyridine | ...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.51E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8894 (3-(3-Methyl-3,4-dihydronaphthalen-2-yl)pyridine | ...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.79E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8910 (3-(5-Chloro-6-methoxy-2-naphthyl)pyridine | 3-(5-c...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.81E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8916 (1-(2-Naphthyl)-1H-imidazole | 1-(naphthalen-2-yl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 2.82E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8895 (3-(4-Methyl-3,4-dihydronaphthalen-2-yl)pyridine | ...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.55E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8904 (3-(2-Naphthyl)pyridine | 3-(naphthalen-2-yl)pyridi...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 5.73E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8892 (3-(1-Methyl-3,4-dihydronaphthalen-2-yl)-pyridine |...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 6.05E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8908 (3-(6-Ethoxy-2-naphthyl)pyridine | 3-(6-ethoxynapht...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.64E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM8911 (3-(5-Bromo-6-methoxy-2-naphthyl)pyridine | 3-(5-br...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.11E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
UNIVERSITAT DES SAARLANDES US Patent | Assay Description The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th... | US Patent US9271963 (2016) BindingDB Entry DOI: 10.7270/Q2445KBN | |||||||||||
More data for this Ligand-Target Pair |