Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359846 (CHEMBL1233807) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM34038 (4,5,6,7-tetraiodobenzimidazole (TIBI), 1a) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359842 (CHEMBL1928905) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359840 (CHEMBL1928903) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50156680 (2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359841 (CHEMBL1928904) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50156673 (((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359843 (CHEMBL1928906) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359847 (CHEMBL1928909) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 93 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM34053 (iodinated benzimidazole, 16) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 106 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50156670 (2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 133 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359845 (CHEMBL1928908) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 195 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM34055 (iodinated benzimidazole, 21) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 324 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM34059 (brominated benzimidazole, 20) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MMDB PC cid PC sid PDB UniChem | Article PubMed | 342 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50156669 (4,5,6,7-TETRABROMO-BENZIMIDAZOLE | 4,5,6,7-tetrabr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 343 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha' (Homo sapiens (Human)) | BDBM50359844 (CHEMBL1928907) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 768 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The John Paul II Catholic University of Lublin Curated by ChEMBL | Assay Description Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ... | Eur J Med Chem 47: 345-50 (2012) Article DOI: 10.1016/j.ejmech.2011.11.002 BindingDB Entry DOI: 10.7270/Q2377944 | |||||||||||
More data for this Ligand-Target Pair |