Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18193 (1-ethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinoli...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 8.10E+3 | -27.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 4 |
Ligand Pharmaceuticals Inc. | Assay Description The procedure for the cross reactivity receptor binding assays was using baculovirus-expressed receptors. After correcting for nonspecific binding, I... | J Med Chem 50: 2486-96 (2007) Article DOI: 10.1021/jm061329j BindingDB Entry DOI: 10.7270/Q20R9MNK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18198 (1-(cyclopropylmethyl)-9-(trifluoromethyl)-1H,2H,3H...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 8.80E+3 | -26.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 4 |
Ligand Pharmaceuticals Inc. | Assay Description The procedure for the cross reactivity receptor binding assays was using baculovirus-expressed receptors. After correcting for nonspecific binding, I... | J Med Chem 50: 2486-96 (2007) Article DOI: 10.1021/jm061329j BindingDB Entry DOI: 10.7270/Q20R9MNK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18197 (1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 9.20E+3 | -26.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 4 |
Ligand Pharmaceuticals Inc. | Assay Description The procedure for the cross reactivity receptor binding assays was using baculovirus-expressed receptors. After correcting for nonspecific binding, I... | J Med Chem 50: 2486-96 (2007) Article DOI: 10.1021/jm061329j BindingDB Entry DOI: 10.7270/Q20R9MNK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141381 (US8916600, 15 | US8916600, 16 | US9738632, Example...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.64 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141381 (US8916600, 15 | US8916600, 16 | US9738632, Example...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.27 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141383 (US8916600, 17 | US9738632, Example 17) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.996 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141384 (US8916600, 18 | US9738632, Example 18) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.44 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141385 (US8916600, 19 | US9738632, Example 19) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.663 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM141386 (US8916600, 20 | US9738632, Example 20) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.96 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Astrazeneca AB; Bayer Pharma Aktiengesellschaft US Patent | Assay Description In the GR radioligand binding assay, test compounds were serially diluted in semi-log steps (10 concentrations) with a final concentration of 10 uM. ... | US Patent US8916600 (2014) BindingDB Entry DOI: 10.7270/Q2WQ02HG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18702 (dihydroquinoline compound, 14 | {[6-(2-methoxyphen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18704 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-en-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18705 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-en-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18706 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(propylsulfany...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.02E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18707 (4-[(cyclopentylsulfanyl)methyl]-6-(2-methoxyphenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 548 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18708 (4-[(cyclohexylsulfanyl)methyl]-6-(2-methoxyphenyl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 371 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18709 (6-(2-methoxyphenyl)-2,2-dimethyl-4-{[(2-methylbuty...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 303 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18710 (6-(2-methoxyphenyl)-2,2-dimethyl-4-{[(3-methylbuty...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 703 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18711 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(phenylsulfany...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 804 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18712 (4-[(benzylsulfanyl)methyl]-6-(2-methoxyphenyl)-2,2...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18713 (6-(2-methoxyphenyl)-2,2-dimethyl-4-{[(2-phenylethy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 194 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18714 (4-{[(4-chlorophenyl)sulfanyl]methyl}-6-(2-methoxyp...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18715 (1-({[6-(2-methoxyphenyl)-2,2-dimethyl-1,2-dihydroq...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18716 (6-(2-methoxyphenyl)-2,2,4-trimethyl-1,2-dihydroqui...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18717 (6-(2-fluorophenyl)-2,2-dimethyl-4-[(prop-2-en-1-yl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18718 (6-(3-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-en-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18719 (6-(5-fluoro-2-methoxyphenyl)-2,2-dimethyl-4-[(prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18720 (2-chloro-3-{2,2-dimethyl-4-[(prop-2-en-1-ylsulfany...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 129 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18721 (6-(5-fluoro-2-methoxyphenyl)-2,2-dimethyl-4-{[(2-p...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 84 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18722 (2-chloro-3-(2,2-dimethyl-4-{[(2-phenylethyl)sulfan...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 16: 1549-52 (2006) Article DOI: 10.1016/j.bmcl.2005.12.043 BindingDB Entry DOI: 10.7270/Q25B00RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18724 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-ene-1-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18705 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-en-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18725 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(prop-2-en-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 116 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18704 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[(prop-2-en-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18727 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(prop-2-en-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 116 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18728 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(prop-2-en-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 355 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18729 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[2-methyl-1-(pr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 710 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18730 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(prop-2-en-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18731 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(prop-2-en-1...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18732 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[phenyl(prop-2-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18733 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[2-phenyl-1-(pr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18734 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[3-phenyl-1-(pr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18735 (4-(1-methoxyethyl)-6-(2-methoxyphenyl)-2,2-dimethy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.06E+3 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18736 (4-{1-[(2E)-but-2-en-1-yloxy]ethyl}-6-(2-methoxyphe...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18737 (6-(2-methoxyphenyl)-2,2-dimethyl-4-{1-[(3-methylbu...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 395 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18738 (6-(2-methoxyphenyl)-2,2-dimethyl-4-{1-[(2E)-pent-2...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 565 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18739 (6-(2-methoxyphenyl)-2,2-dimethyl-4-(1-{[(2E)-3-phe...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 980 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18740 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(3-phenylpro...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18741 (6-(2-methoxyphenyl)-2,2-dimethyl-4-[1-(2-phenyleth...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 405 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18742 (4-{1-[2-(2-chlorophenyl)ethoxy]ethyl}-6-(2-methoxy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM18743 (4-{1-[2-(3-chlorophenyl)ethoxy]ethyl}-6-(2-methoxy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 275 | n/a | n/a | n/a | n/a | 7.4 | 22 |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description IC50 values shown are means of a single experiment done in duplicate 11-point concentration-effect curves. | Bioorg Med Chem Lett 17: 5091-5 (2007) Article DOI: 10.1016/j.bmcl.2007.07.021 BindingDB Entry DOI: 10.7270/Q21J981M | |||||||||||
More data for this Ligand-Target Pair |
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