Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM18129 ((2S)-2-amino-3-(4-hydroxyphenyl)propanoic acid | L...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 2.50E+4 | -27.3 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM36555 (3-Aminotyrosine) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 2.00E+5 | -22.0 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM36556 (3-Azidotyrosine) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.00E+5 | -22.0 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM36557 (3-Formyltyrosine) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.00E+5 | -20.9 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM36554 (3-Nitrotyrosine) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 4.00E+5 | -20.2 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin--tyrosine ligase (Homo sapiens (Human)) | BDBM36558 (4-Aminophenylalanine) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents | Article PubMed | >4.00E+6 | >-14.2 | n/a | n/a | n/a | n/a | n/a | 6.8 | 37 |
Binghamton University | Assay Description Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL). | ACS Chem Biol 5: 777-85 (2010) Article DOI: 10.1021/cb100060v BindingDB Entry DOI: 10.7270/Q25H7DM1 | |||||||||||
More data for this Ligand-Target Pair |