Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-dependent protein kinase type I-alpha regulatory subunit (Bos taurus) | BDBM50011236 (CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-dependent protein kinase type I-alpha regulatory subunit (Bos taurus) | BDBM92674 (Isoquinolinesulfonamide, CKI-7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 5.50E+5 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-dependent protein kinase type I-alpha regulatory subunit (Bos taurus) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair |