Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64564 (US9428505, Compound 8) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 3.60E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64562 (US9428505, Compound 7) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 4.10E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64569 (US9428505, Comparative: Example 1) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 4.80E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64551 (US9428505, Compound 1) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5.80E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64555 (US9428505, Compound 3) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 7.20E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64557 (US9428505, Compound 4) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 7.40E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64559 (US9428505, Compound 5) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 8.10E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64575 (US9428505, Comparative: Example 3) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 9.00E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64561 (US9428505, Compound 6) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 9.00E+3 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64567 (US9428505, Compound 11) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64565 (US9428505, Compound 9) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.20E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64570 (US9428505, Comparative: Example 2) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.30E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64553 (US9428505, Compound 2) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.40E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64566 (US9428505, Compound 10) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 2.10E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64578 (US9428505, Comparative: Example 5) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.50E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64579 (US9428505, Comparative: Example 6) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 3.20E+4 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Parathyroid hormone [32-65] (Homo sapiens (Human)) | BDBM64577 (US9428505, Comparative: Example 4) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | 7.4 | n/a |
Chugai Seiyaku Kabushiki Kaisha US Patent | Assay Description HKRK-B7 or LLC-PK1 cells were seeded into a 96-well plate at 1×105 cells/well and incubated overnight. On the following day, 50 μl of cAMP assay... | US Patent US9428505 (2016) BindingDB Entry DOI: 10.7270/Q2VQ31KS | |||||||||||
More data for this Ligand-Target Pair |