Compile Data Set for Download or QSAR

Found 152 hits of ec50 data for polymerid = 340   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526477 (US11186566, Compound 16) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(F)c2)-n2ccc(OCC3C(C)(C)C3(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526510 (US11186566, Compound 49) Show SMILES COc1cccc(c1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526467 (US11186566, Compound 4) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2C)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526476 (US11186566, Compound 15) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2C)-n2ccc(OCC3C(C)(C)C3(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526511 (US11186566, Compound 50) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2F)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526492 (US11186566, Compound 31) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccc(O)cc2)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526489 (US11186566, Compound 28) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(C)c2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526484 (US11186566, Compound 23) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2C)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526464 (US11186566, Compound 1 | US11186566, Compound 17) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526514 (US11186566, Compound 53) Show SMILES COc1ccccc1S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526471 (US11186566, Compound 10) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3(CCC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526475 (US11186566, Compound 14) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526493 (US11186566, Compound 32) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2nc(OCCC3(CC3)C(F)(F)F)cc2F)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526512 (US11186566, Compound 51) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(F)c2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526503 (US11186566, Compound 42) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCCC(C3CC3)C3CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526504 (US11186566, Compound 43) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2Cl)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526523 (US11186566, Compound 63 | US11186566, Compound 64) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C4(CC4)C33CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526519 (US11186566, Compound 58) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2C)-n2ccc(OCC3(CCC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526468 (US11186566, Compound 5) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(F)c2)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526516 (US11186566, Compound 55) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	50	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526526 (US11186566, Compound A) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccnc2N)-n2ccc(OCC(C)(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	60	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526502 (US11186566, Compound 41) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC(C3CC3)C3CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	70	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526500 (US11186566, Compound 39) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(O[C@H]3C[C@H]4CC[C@@H]3C4)n2)C(C)(C)C1 |r,THB:26:27:33:30.31| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	70	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526485 (US11186566, Compound 24) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccc(C)cc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	70	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526498 (US11186566, Compound 37) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(COCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	70	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526501 (US11186566, Compound 40) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C[C@@H]4CC[C@@H]3C4)n2)C(C)(C)C1 |r,THB:27:28:31.32:34| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	80	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526494 (US11186566, Compound 33) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccc(O)cc2)-n2ccc(OCC3C(C)(C)C3(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	80	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526518 (US11186566, Compound 57) Show SMILES COc1ccc(c(C)c1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	80	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526491 (US11186566, Compound 30 | US11186566, Compound 36) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C(C)(C)C3(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	90	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526507 (US11186566, Compound 46) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)N[S@@](=N)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526504 (US11186566, Compound 43) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2Cl)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526510 (US11186566, Compound 49) Show SMILES COc1cccc(c1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526511 (US11186566, Compound 50) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2F)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526512 (US11186566, Compound 51) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(F)c2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526513 (US11186566, Compound 52) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccc(F)cc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526514 (US11186566, Compound 53) Show SMILES COc1ccccc1S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526515 (US11186566, Compound 54) Show SMILES COc1ccc(cc1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526516 (US11186566, Compound 55) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526518 (US11186566, Compound 57) Show SMILES COc1ccc(c(C)c1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526519 (US11186566, Compound 58) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2C)-n2ccc(OCC3(CCC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526520 (US11186566, Compound 59) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2cccc(F)c2)-n2ccc(OCC3(CCC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526523 (US11186566, Compound 63 | US11186566, Compound 64) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C4(CC4)C33CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526508 (US11186566, Compound 47) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)N[S@](=N)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526503 (US11186566, Compound 42) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCCC(C3CC3)C3CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526502 (US11186566, Compound 41) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC(C3CC3)C3CC3)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526501 (US11186566, Compound 40) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C[C@@H]4CC[C@@H]3C4)n2)C(C)(C)C1 |r,THB:27:28:31.32:34| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526500 (US11186566, Compound 39) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(O[C@H]3C[C@H]4CC[C@@H]3C4)n2)C(C)(C)C1 |r,THB:26:27:33:30.31| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526498 (US11186566, Compound 37) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(COCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526491 (US11186566, Compound 30 | US11186566, Compound 36) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3C(C)(C)C3(C)C)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480] (Homo sapiens (Human))	BDBM526464 (US11186566, Compound 1 | US11186566, Compound 17) Show SMILES C[C@@H]1CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCCC3(CC3)C(F)(F)F)n2)C(C)(C)C1 |r| Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	<100	n/a	n/a	n/a	n/a
TBA					Assay Description The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...				Citation and Details BindingDB Entry DOI: 10.7270/Q22R3VVH
					More data for this Ligand-Target Pair

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