Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM86143 (L-Val-L-Pro-L-Asn-L-Leu-L-Pro-L-Gln-L-Arg-L-Phe-NH...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50029138 (CHEMBL3360830) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
The University of Mississippi Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor | J Med Chem 57: 8903-27 (2014) Article DOI: 10.1021/jm500989n BindingDB Entry DOI: 10.7270/Q2C24Z18 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50037557 (2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human NPFFR2 expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cyclic cAMP accumulation | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50565182 (CHEMBL4797394) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human NPFFR2 expressed in CHO cells by [35S]-GTP S binding assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555154 (CHEMBL4800237) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555154 (CHEMBL4800237) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50565181 (CHEMBL4783555) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK-293A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50037557 (2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Lanzhou University Curated by ChEMBL | Assay Description Agonist activity at NPFF2 receptor (unknown origin) expressed in HEK293A cells assessed as inhibition of forskolin-stimulated cAMP accumulation measu... | Bioorg Med Chem 27: 630-643 (2019) Article DOI: 10.1016/j.bmc.2019.01.003 BindingDB Entry DOI: 10.7270/Q2M61PJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558732 (CHEMBL4759079) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 41 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50037557 (2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 42 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558732 (CHEMBL4759079) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 42 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50037557 (2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 43 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581384 (CHEMBL5085455) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581384 (CHEMBL5085455) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581386 (CHEMBL5085013) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 81 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581386 (CHEMBL5085013) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 82 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558728 (CHEMBL4777803) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 87 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558728 (CHEMBL4777803) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 87 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50565186 (CHEMBL4785076) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in mouse NIH3T3 cells by receptor selection and amplification technology assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50414854 (CHEMBL574565) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
ACADIA Pharmaceuticals AB Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 days | J Med Chem 52: 6511-4 (2009) Article DOI: 10.1021/jm9011998 BindingDB Entry DOI: 10.7270/Q2G73FZF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50414852 (CHEMBL573738) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
ACADIA Pharmaceuticals AB Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 days | J Med Chem 52: 6511-4 (2009) Article DOI: 10.1021/jm9011998 BindingDB Entry DOI: 10.7270/Q2G73FZF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581385 (CHEMBL5086601) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 112 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581385 (CHEMBL5086601) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 112 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555153 (CHEMBL4744365) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555153 (CHEMBL4744365) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50414856 (CHEMBL573519) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 126 | n/a | n/a | n/a | n/a |
ACADIA Pharmaceuticals AB Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 days | J Med Chem 52: 6511-4 (2009) Article DOI: 10.1021/jm9011998 BindingDB Entry DOI: 10.7270/Q2G73FZF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50553312 (CHEMBL4745052) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
TBA | Assay Description Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence... | Citation and Details Article DOI: 10.1021/acsmedchemlett.9b00182 BindingDB Entry DOI: 10.7270/Q2VM4GX0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558734 (CHEMBL4755334) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 132 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558734 (CHEMBL4755334) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 132 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581388 (CHEMBL5094675) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 132 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581388 (CHEMBL5094675) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 133 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50553312 (CHEMBL4745052) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
TBA | Assay Description Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence... | Citation and Details Article DOI: 10.1021/acsmedchemlett.9b00182 BindingDB Entry DOI: 10.7270/Q2VM4GX0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50553308 (CHEMBL4742191) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
TBA | Assay Description Activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence... | Citation and Details Article DOI: 10.1021/acsmedchemlett.9b00182 BindingDB Entry DOI: 10.7270/Q2VM4GX0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50565183 (CHEMBL4790994) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 157 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human NPFFR2 expressed in CHO cells by [35S]-GTP S binding assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50508423 (CHEMBL4449491) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
Lanzhou University Curated by ChEMBL | Assay Description Agonist activity at NPFF2 receptor (unknown origin) expressed in HEK293A cells assessed as inhibition of forskolin-stimulated cAMP accumulation measu... | Bioorg Med Chem 27: 630-643 (2019) Article DOI: 10.1016/j.bmc.2019.01.003 BindingDB Entry DOI: 10.7270/Q2M61PJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50414855 (CHEMBL573518) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
ACADIA Pharmaceuticals AB Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in cells assessed as beta-galactosidase levels after 5 days | J Med Chem 52: 6511-4 (2009) Article DOI: 10.1021/jm9011998 BindingDB Entry DOI: 10.7270/Q2G73FZF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555155 (CHEMBL4788060) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 168 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555155 (CHEMBL4788060) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50508423 (CHEMBL4449491) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a |
Lanzhou University Curated by ChEMBL | Assay Description Agonist activity at NPFF2 receptor (unknown origin) expressed in HEK293A cells assessed as inhibition of forskolin-stimulated cAMP accumulation measu... | Bioorg Med Chem 27: 630-643 (2019) Article DOI: 10.1016/j.bmc.2019.01.003 BindingDB Entry DOI: 10.7270/Q2M61PJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555148 (CHEMBL4745148) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 178 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human NPFFR2 expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by LANCE ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555148 (CHEMBL4745148) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555148 (CHEMBL4745148) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558730 (CHEMBL4792870) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50558730 (CHEMBL4792870) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 186 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555148 (CHEMBL4745148) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 186 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30... | Citation and Details BindingDB Entry DOI: 10.7270/Q2TQ657S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555148 (CHEMBL4745148) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 186 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581387 (CHEMBL5086463) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50581387 (CHEMBL5086463) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 191 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00694 BindingDB Entry DOI: 10.7270/Q2VM4H43 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555156 (CHEMBL4750006) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 191 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50555156 (CHEMBL4750006) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 192 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01367 BindingDB Entry DOI: 10.7270/Q2NG4V97 | |||||||||||
More data for this Ligand-Target Pair |
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