Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250673 (US9447148, 9.42 | US9447148, 9.55) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00200 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250673 (US9447148, 9.42 | US9447148, 9.55) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00200 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250661 (US9447148, 9.30) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00200 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250668 (US9447148, 9.37 | US9447148, 9.50) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00300 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250649 (US9447148, 9.18) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00300 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250668 (US9447148, 9.37 | US9447148, 9.50) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00300 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250648 (US9447148, 9.17) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250642 (US9447148, 9.10) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50590037 (CHEMBL5191309) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00793 BindingDB Entry DOI: 10.7270/Q20C50R5 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250653 (US9447148, 9.22) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250652 (US9447148, 9.21) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250651 (US9447148, 9.20) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00400 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250643 (US9447148, 9.11) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00500 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM135768 (US10179804, Example 153 | US10632171, Peptide No. ...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 0.00500 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM82411 (CAS_75921-69-6 | NDP-MSH) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.00500 | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Decrease in frog skin reflectivity (melanotropic activity). | J Med Chem 40: 2740-9 (1997) Article DOI: 10.1021/jm970018t BindingDB Entry DOI: 10.7270/Q2057GKD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50033130 ((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0.00500 | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluated for agonist activity against human Melanocortin 1 receptor using hMC1-R assay | J Med Chem 38: 3454-61 (1995) BindingDB Entry DOI: 10.7270/Q2Z32094 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50033130 ((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0.00500 | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluated for agonist activity at cloned mammalian human MSH1 receptor | J Med Chem 38: 3454-61 (1995) BindingDB Entry DOI: 10.7270/Q2Z32094 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250660 (US9447148, 9.29) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250655 (US9447148, 9.24) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ... | Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00561 BindingDB Entry DOI: 10.7270/Q2N301KK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250671 (US9447148, 9.40 | US9447148, 9.53) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250634 (US9447148, 9.2 | US9447148, 9.31) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250671 (US9447148, 9.40 | US9447148, 9.53) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00600 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250659 (US9447148, 9.28) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00700 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250654 (US9447148, 9.23) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00700 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250633 (US9447148, 9.1) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00700 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250672 (US9447148, 9.41 | US9447148, 9.54) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00800 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250641 (US9447148, 9.9) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00800 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250672 (US9447148, 9.41 | US9447148, 9.54) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00800 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250635 (US9447148, 9.3) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00800 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50121900 (Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.00800 | n/a | n/a | n/a | n/a |
The Hebrew University of Jerusalem Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells | J Med Chem 51: 1026-34 (2008) Article DOI: 10.1021/jm701093y BindingDB Entry DOI: 10.7270/Q29W0GC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50590040 (CHEMBL5185945) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | <0.00900 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00793 BindingDB Entry DOI: 10.7270/Q20C50R5 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50131251 ((S)-5-Guanidino-2-{(S)-2-[(S)-3-(3H-imidazol-4-yl)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0.00900 | n/a | n/a | n/a | n/a |
University of Cincinnati Curated by ChEMBL | Assay Description Binding affinity towards human melanocortin 4 receptor (hMC4R) | Bioorg Med Chem Lett 13: 2647-50 (2003) BindingDB Entry DOI: 10.7270/Q2474BD9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50152246 ((S)-5-Guanidino-2-((S)-2-{(S)-2-[(S)-3-(3H-imidazo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.00900 | n/a | n/a | n/a | n/a |
University of Cincinnati Curated by ChEMBL | Assay Description Agonistic activity against against human Melanocortin 1 receptor | Bioorg Med Chem Lett 14: 4839-42 (2004) Article DOI: 10.1016/j.bmcl.2004.07.046 BindingDB Entry DOI: 10.7270/Q2445KX8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250658 (US9447148, 9.27) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.00900 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50590040 (CHEMBL5185945) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >0.00912 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00793 BindingDB Entry DOI: 10.7270/Q20C50R5 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50033130 ((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0.00950 | n/a | n/a | n/a | n/a |
University of Arizona Curated by ChEMBL | Assay Description Evaluated for agonist activity against mouse Melanocortin 1 receptor using mMC1R assay | J Med Chem 38: 3454-61 (1995) BindingDB Entry DOI: 10.7270/Q2Z32094 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50301155 (CHEMBL569693 | Ph(CH2)3CO-His-D-Phe-Arg-Trp-NH2) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | n/a | n/a |
University of Cincinnati Curated by ChEMBL | Assay Description Agonistic activity against human MC1R | Bioorg Med Chem Lett 19: 5176-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.025 BindingDB Entry DOI: 10.7270/Q2WD41JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells incubated for 2 hrs by AlphaScreen cAMP assay | J Med Chem 61: 7729-7740 (2018) Article DOI: 10.1021/acs.jmedchem.8b00684 BindingDB Entry DOI: 10.7270/Q2X63QHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ... | J Med Chem 63: 2194-2208 (2020) Article DOI: 10.1021/acs.jmedchem.9b00860 BindingDB Entry DOI: 10.7270/Q25142KG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50250586 (CHEMBL4093140) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | n/a | n/a |
The University of Arizona Curated by ChEMBL | Assay Description Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting method | J Med Chem 60: 9320-9329 (2017) Article DOI: 10.1021/acs.jmedchem.7b01295 BindingDB Entry DOI: 10.7270/Q2XG9TJB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse MC1R by alphascreen cAMP assay | Citation and Details Article DOI: 10.1021/acsmedchemlett.9b00641 BindingDB Entry DOI: 10.7270/Q2VQ36C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250645 (US9447148, 9.13) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.0100 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250647 (US9447148, 9.15) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.0120 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0120 | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ... | ACS Med Chem Lett 11: 272-277 (2020) Article DOI: 10.1021/acsmedchemlett.9b00198 BindingDB Entry DOI: 10.7270/Q2QV3QTB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0120 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as induction of cAMP level at 100 uM incubated for 2 hr by alphaScreen assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01417 BindingDB Entry DOI: 10.7270/Q2RR231G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250638 (US9447148, 9.6) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.0140 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50121900 (Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0140 | n/a | n/a | n/a | n/a |
University of Cincinnati Curated by ChEMBL | Assay Description Agonistic activity against mouse MC1R | Bioorg Med Chem Lett 19: 5176-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.025 BindingDB Entry DOI: 10.7270/Q2WD41JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Mus musculus) | BDBM50017181 (CHEMBL441738) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0150 | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Agonist activity at mouse MC1R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ... | J Med Chem 60: 805-813 (2017) Article DOI: 10.1021/acs.jmedchem.6b01707 BindingDB Entry DOI: 10.7270/Q2R213MT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM250644 (US9447148, 9.12) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.0150 | n/a | n/a | 7.5 | 37 |
Palatin Technologies, Inc. US Patent | Assay Description Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ... | US Patent US9447148 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HD2 | |||||||||||
More data for this Ligand-Target Pair |
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