Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543473 ((((6-chloro-5-(2'-hydroxy-[1,1'-biphenyl]-4- yl)-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.550 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543471 ((((6-chloro-5-(2'-hydroxy-[1,1'-biphenyl]-4- yl)-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.970 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543477 (2-((6-chloro-5-(2'-hydroxy-4'-(1H-1,2,4- triazol-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192505 (US9187477, 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.20 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543470 (2-((6-chloro-5-(2'-hydroxy-[1,1'-biphenyl]-4- yl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543472 (US11279702, Compound 3 | ethyl hydrogen (((6-chlor...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.38 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201005 (US9540364, example 15) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 3 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201004 (US9540364, example 14) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 4 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201001 (US9540364, example 13) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200996 (US9540364, example 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201006 (US9540364, example 16) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 6 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192510 (US9187477, 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 6 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200995 (US9540364, example 7) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 8 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200992 (US9540364, example 3) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 8 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192508 (US9187477, 16 | US9187477, 4) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 12 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192513 (US9187477, 9) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 17 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543476 (2-((5-(4'-(1H-1,2,4-triazol-1-yl)-[1,1'- biphenyl]...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201007 (US9540364, example 17) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 20 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192514 (US9187477, 10) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 26 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192506 (US9187477, 2) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 32 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200997 (US9540364, example 9) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 33 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201008 (US9540364, example 18) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 34 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200998 (US9540364, example 10) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 34 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192515 (US9187477, 11) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 35 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201011 (US9540364, example 21) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 38 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543475 ((S)-2-((6-chloro-5-(4-(3-hydroxypyrrolidin- 1-yl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 43 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201010 (US9540364, example 20) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 50 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM201009 (US9540364, example 19) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 67 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200999 (US9540364, example 12) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 76 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200993 (US9540364, example 4) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 104 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192507 (US9187477, 3) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 108 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Rattus norvegicus) | BDBM50242401 (4-hydroxy-3-(2'-hydroxybiphenyl-4-yl)-6-oxo-6,7-di...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 116 | n/a | n/a | n/a | n/a |
Lund University Curated by ChEMBL | Assay Description Activation of rat AMPKalpha1alpha2beta1gamma1 kinase | J Biol Chem 282: 32549-60 (2007) Article DOI: 10.1074/jbc.M706536200 BindingDB Entry DOI: 10.7270/Q2BC3ZBQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192509 (US9187477, 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 119 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192519 (US9187477, 15) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 133 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543469 (US11279702, Compound A1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200994 (US9540364, example 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 209 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200907 (US9540364, example 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | n/a | n/a | 216 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192508 (US9187477, 16 | US9187477, 4) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 290 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192512 (US9187477, 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 339 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192511 (US9187477, 7) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 468 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192518 (US9187477, 14) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 578 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM543474 (2-((6-chloro-5-(4'-(3,3-dimethylbutyl)-2'- hydroxy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.12E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2XW4P0R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192516 (US9187477, 12) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.31E+3 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM192517 (US9187477, 13) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 2.04E+3 | n/a | n/a | 7.0 | n/a |
Boehringer Ingelheim International GmbH US Patent | Assay Description Activated AMPK complex 1 (containing alphal betalgammal ) was obtained from baculovirus expression system. The gene encoding AMPK alphal was cloned i... | US Patent US9187477 (2015) BindingDB Entry DOI: 10.7270/Q2CR5S58 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM50434271 (CHEMBL2385951) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Activation of recombinant AMPK alpha1 (1 to 394) (unknown origin) after 2 hrs by scintillation proximity assay | ACS Med Chem Lett 4: 475-80 (2013) Article DOI: 10.1021/ml400028q BindingDB Entry DOI: 10.7270/Q2Z039HW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM200991 (US9540364, example 2) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 4.29E+3 | n/a | n/a | 7.3 | n/a |
Merck Sharp & Dohme Corp. US Patent | Assay Description The in vitro AMPK activation assay is performed in a volume of 30 μl in a 384-well plate. Enzyme reactions were assembled in the microtiter plat... | US Patent US9540364 (2017) BindingDB Entry DOI: 10.7270/Q2SB43X2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM50434272 (CHEMBL1242297) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of human recombinant AMPK alpha1 (1 to 394 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL using SAMS peptide after 10 m... | Bioorg Med Chem Lett 26: 5139-5148 (2016) Article DOI: 10.1016/j.bmcl.2016.09.065 BindingDB Entry DOI: 10.7270/Q25M67PH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM50434272 (CHEMBL1242297) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a |
University of Nebraska Medical Center Curated by ChEMBL | Assay Description Activation of human recombinant AMPK alpha1 subunit | J Med Chem 58: 2-29 (2015) Article DOI: 10.1021/jm401994c BindingDB Entry DOI: 10.7270/Q2KH0PZW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM50434272 (CHEMBL1242297) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Activation of human AMPK alpha1 (1 to 394) expressed in African green monkey COS7 cells | ACS Med Chem Lett 4: 475-80 (2013) Article DOI: 10.1021/ml400028q BindingDB Entry DOI: 10.7270/Q2Z039HW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5'-AMP-activated protein kinase catalytic subunit alpha-1 (Homo sapiens (Human)) | BDBM50434272 (CHEMBL1242297) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Activation of recombinant AMPK alpha1 (1 to 394) (unknown origin) after 2 hrs by scintillation proximity assay | ACS Med Chem Lett 4: 475-80 (2013) Article DOI: 10.1021/ml400028q BindingDB Entry DOI: 10.7270/Q2Z039HW | |||||||||||
More data for this Ligand-Target Pair |