Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Axin-2 (Homo sapiens (Human)) | BDBM50318567 (2-(4-(Trifluoromethyl)phenyl)-7,8-dihydro-5H-thiop...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 371 | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Stabilization of Axin2 in human SW480 cells after 24 hrs by sandwich ELISA | J Med Chem 55: 1127-36 (2012) Article DOI: 10.1021/jm2011222 BindingDB Entry DOI: 10.7270/Q2BK1DCV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Axin-2 (Homo sapiens (Human)) | BDBM50380595 (CHEMBL1867804) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 375 | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Stabilization of Axin2 in human SW480 cells after 24 hrs by sandwich ELISA | J Med Chem 55: 1127-36 (2012) Article DOI: 10.1021/jm2011222 BindingDB Entry DOI: 10.7270/Q2BK1DCV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Axin-2 (Homo sapiens (Human)) | BDBM50380592 (CHEMBL1552719) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 566 | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Stabilization of Axin2 in human SW480 cells after 24 hrs by sandwich ELISA | J Med Chem 55: 1127-36 (2012) Article DOI: 10.1021/jm2011222 BindingDB Entry DOI: 10.7270/Q2BK1DCV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Axin-2 (Homo sapiens (Human)) | BDBM50380590 (CHEMBL1898239) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 709 | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Stabilization of Axin2 in human SW480 cells after 24 hrs by sandwich ELISA | J Med Chem 55: 1127-36 (2012) Article DOI: 10.1021/jm2011222 BindingDB Entry DOI: 10.7270/Q2BK1DCV | |||||||||||
More data for this Ligand-Target Pair |