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Compile Data Set for Download or QSAR

Found 1 hit of ec50 data for polymerid = 50006480   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transient receptor potential cation channel subfamily M member 8


(Mus musculus)		BDBM50329105
PNG
(19(S)-Heyneanine | CHEMBL463317 | voacristine)
Show SMILES COC(=O)[C@@]12C[C@@H]3C[C@H]([C@H](C)O)[C@@H]1N(C3)CCc1c2[nH]c2ccc(OC)cc12 |r,TLB:8:12:18.17.16.15:5.6.14,9:8:4.5:13.14|
Show InChI InChI=1S/C22H28N2O4/c1-12(25)16-8-13-10-22(21(26)28-3)19-15(6-7-24(11-13)20(16)22)17-9-14(27-2)4-5-18(17)23-19/h4-5,9,12-13,16,20,23,25H,6-8,10-11H2,1-3H3/t12-,13-,16+,20-,22+/m0/s1
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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 2.70E+4n/an/an/an/a



University of Shizuoka

Curated by ChEMBL


Assay Description
Agonist activity at mouse TRPM8 expressed in T-REx HEK cells assessed as increase in intracellular Ca2+ accumulation by Fluo-4 AM dye based fluoresce...

J. Nat. Prod. 77: 1831-8 (2014)


Article DOI: 10.1021/np500235b
BindingDB Entry DOI: 10.7270/Q27S7QDF
More data for this
Ligand-Target Pair