Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581658 (CHEMBL5092307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.5 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581658 (CHEMBL5092307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581650 (CHEMBL5081975) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581650 (CHEMBL5081975) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.5 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581654 (CHEMBL5082551) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581654 (CHEMBL5082551) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603315 (CHEMBL5202580) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581655 (CHEMBL5080998) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581655 (CHEMBL5080998) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581658 (CHEMBL5092307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581658 (CHEMBL5092307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581657 (CHEMBL5088494) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 64 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581657 (CHEMBL5088494) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 65 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581650 (CHEMBL5081975) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 134 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581650 (CHEMBL5081975) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 135 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581657 (CHEMBL5088494) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581657 (CHEMBL5088494) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 151 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603324 (CHEMBL5174724) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603322 (CHEMBL5203480) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581651 (CHEMBL5077507) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 195 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581651 (CHEMBL5077507) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 195 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603320 (CHEMBL5200919) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603326 (CHEMBL5170854) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603327 (CHEMBL5202223) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581652 (CHEMBL5085505) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517133 (CHEMBL4448632) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581652 (CHEMBL5085505) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 282 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603319 (CHEMBL5192437) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603316 (CHEMBL5190234) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603321 (CHEMBL5183095) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517152 (CHEMBL4527534) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 430 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603323 (CHEMBL5180985) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 440 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50603325 (CHEMBL5185986) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 450 | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmc.2021.116587 BindingDB Entry DOI: 10.7270/Q28W3JCR | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517131 (CHEMBL4472664) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 510 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581656 (CHEMBL5082981) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 513 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581656 (CHEMBL5082981) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 513 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581653 (CHEMBL5089041) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 562 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581653 (CHEMBL5089041) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 564 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517138 (CHEMBL4557657) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 940 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581656 (CHEMBL5082981) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 955 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50581656 (CHEMBL5082981) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 966 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01804 BindingDB Entry DOI: 10.7270/Q24X5CN4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517151 (CHEMBL4467290) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517147 (CHEMBL4575422) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517130 (CHEMBL4476788) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517128 (CHEMBL4448308) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517126 (CHEMBL4463797) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517146 (CHEMBL4561076) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517125 (CHEMBL4474605) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517150 (CHEMBL4538515) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chemerin-like receptor 1 (Homo sapiens (Human)) | BDBM50517135 (CHEMBL4472121) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a |
Kyowa Kirin Co., Ltd. Curated by ChEMBL | Assay Description Agonist activity at chemR23 expressed in human CAL1 cells assessed as increase in intracellular calcium ion concentration | Bioorg Med Chem 27: (2019) Article DOI: 10.1016/j.bmc.2019.115091 BindingDB Entry DOI: 10.7270/Q2N30190 | |||||||||||
More data for this Ligand-Target Pair |
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