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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
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Ki
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Compile Data Set for Download or QSAR
Found
114
hits of ec50 data for polymerid = 50006766
Target/Host
(Institution)
Ligand
Target/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
k
off
s
-1
k
on
M
-1
s
-1
pH
Temp
°C
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571573
(CHEMBL4863993)
Show SMILES
Clc1cnc(CNc2cc3sncc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
7.90
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571573
(CHEMBL4863993)
Show SMILES
Clc1cnc(CNc2cc3sncc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
7.90
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571634
(CHEMBL4877000)
Show SMILES
Cn1c(Cl)cnc1CNc1cc2sncc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
11
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571635
(CHEMBL4856061)
Show SMILES
Cc1cc2cnsc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
18
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571618
(CHEMBL4869759)
Show SMILES
Clc1cnc(CNc2cc3cnsc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
25
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571636
(CHEMBL4855103)
Show SMILES
Fc1cc2cnsc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
29
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571637
(CHEMBL4857667)
Show SMILES
Cc1cc2cnsc2cc1NCc1ncc(Cl)n1C
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
38
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571617
(CHEMBL4860824)
Show SMILES
Cc1cc2sncc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
39
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571572
(CHEMBL4854482)
Show SMILES
Clc1cnc(CNc2ccc3cnsc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
44
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602146
(CHEMBL5177026)
Show SMILES
OC[C@@H]1Cc2cc(Cl)c(Cl)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
50
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602165
(CHEMBL5193084)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
63
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571638
(CHEMBL4845759)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1ccc2cnsc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
85
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571571
(CHEMBL4849726)
Show SMILES
Clc1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
89
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571619
(CHEMBL4873593)
Show SMILES
Fc1cc2sncc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
98
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602162
(CHEMBL5194924)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
100
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571639
(CHEMBL4862183)
Show SMILES
Cn1c(Cl)cnc1CNc1cc2sncc2cc1F
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
102
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602168
(CHEMBL5192928)
Show SMILES
OC[C@H]1Cc2cc(ccc2[C@H](N1)c1cc(F)cc(Cl)c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
125
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602168
(CHEMBL5192928)
Show SMILES
OC[C@H]1Cc2cc(ccc2[C@H](N1)c1cc(F)cc(Cl)c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
126
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571605
(CHEMBL4869736)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
158
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571607
(CHEMBL4863223)
Show SMILES
Cn1c(Cl)cnc1CN(CC1CC1)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
158
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602164
(CHEMBL5186500)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(F)cc(F)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
200
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602163
(CHEMBL5189636)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(Cl)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
200
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602170
(CHEMBL5188072)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1cc(F)cc(c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
251
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571640
(CHEMBL4866122)
Show SMILES
Cn1c(Cl)cnc1CNc1ccc2cnsc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
295
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571641
(CHEMBL4849376)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1cc2sncc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
309
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602148
(CHEMBL5181952)
Show SMILES
OC[C@@H]1Cc2cc(Cl)c(F)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
316
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602160
(CHEMBL5179994)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cccc(F)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
316
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571570
(CHEMBL4876211)
Show SMILES
Cn1c(Cl)cnc1CNc1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
331
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571606
(CHEMBL4863555)
Show SMILES
CN(Cc1ncc(Cl)s1)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
447
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571592
(CHEMBL4855887)
Show SMILES
Cn1c(Br)cnc1CNc1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
457
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571611
(CHEMBL4849797)
Show SMILES
CCN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
468
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571620
(CHEMBL4858854)
Show SMILES
Clc1cnc(CNc2cc3cnsc3cn2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
468
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571598
(CHEMBL4874619)
Show SMILES
FC(F)(F)c1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
490
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602159
(CHEMBL5202815)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cccc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
501
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602147
(CHEMBL5209164)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
501
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571599
(CHEMBL4866780)
Show SMILES
Cc1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
575
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602135
(CHEMBL5209032)
Show SMILES
Cn1c2ccccc2s\c1=N\C(=S)NCC=C
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
631
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602141
(CHEMBL5175850)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
794
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571616
(CHEMBL4867011)
Show SMILES
Clc1cnc(COc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
832
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571623
(CHEMBL4872165)
Show SMILES
Fc1c(NCc2ncc(Cl)s2)ccc2sncc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
933
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602161
(CHEMBL5184410)
Show SMILES
Cc1cc(ccc1Cl)[C@@H]1N[C@H](CO)Cc2ccc(Cl)cc12 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.00E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571624
(CHEMBL4848175)
Show SMILES
Clc1cnc(CNc2ccc3sncc3n2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.18E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602149
(CHEMBL5175871)
Show SMILES
OC[C@@H]1Cc2c(Cl)cccc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.26E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571627
(CHEMBL4855018)
Show SMILES
Fc1cc(NCc2ncc(Cl)s2)cc2cnsc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.38E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571633
(CHEMBL4871607)
Show SMILES
Clc1cnc(CNc2cccc3cnsc23)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.45E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571622
(CHEMBL4861157)
Show SMILES
Clc1cnc(CNc2ccc3sncc3c2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.59E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602158
(CHEMBL5169709)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1ccccc1Cl |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.59E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571629
(CHEMBL4850037)
Show SMILES
CN(Cc1ncc(Cl)s1)c1cc2cnsc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.62E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571621
(CHEMBL4864644)
Show SMILES
Cc1c(NCc2ncc(Cl)s2)ccc2sncc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.74E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602166
(CHEMBL5203756)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ncc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
2.00E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
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