Home
Info
Download
About us
Email us
Contribute data
Web Services
Beta Site
myBDB
logout
Search and Browse
Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
Special tools
3D Structure Series
Find My Compound's Targets
Find Compounds for My Targets
Do Virtual Screening
SCOP
Citation
Author
Journal/Citation
Institution
PubMed
PubChem BioAssay
US Patent
Special Data Sets
D3R
Host Guest Systems
Prot-Lig Validation Sets
Other Databases
PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
Download
All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
Enter Data
Deposition
Contribute data
Sent Comments
Compile Data Set for Download or QSAR
Found
114
hits of ec50 data for polymerid = 50006766,50006766
Target/Host
(Institution)
Ligand
Target/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
k
off
s
-1
k
on
M
-1
s
-1
pH
Temp
°C
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571573
(CHEMBL4863993)
Show SMILES
Clc1cnc(CNc2cc3sncc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
7.90
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571573
(CHEMBL4863993)
Show SMILES
Clc1cnc(CNc2cc3sncc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
7.90
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571634
(CHEMBL4877000)
Show SMILES
Cn1c(Cl)cnc1CNc1cc2sncc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
11
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571635
(CHEMBL4856061)
Show SMILES
Cc1cc2cnsc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
18
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571618
(CHEMBL4869759)
Show SMILES
Clc1cnc(CNc2cc3cnsc3cc2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
25
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571636
(CHEMBL4855103)
Show SMILES
Fc1cc2cnsc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
29
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571637
(CHEMBL4857667)
Show SMILES
Cc1cc2cnsc2cc1NCc1ncc(Cl)n1C
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
38
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571617
(CHEMBL4860824)
Show SMILES
Cc1cc2sncc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
39
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571572
(CHEMBL4854482)
Show SMILES
Clc1cnc(CNc2ccc3cnsc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
44
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602146
(CHEMBL5177026)
Show SMILES
OC[C@@H]1Cc2cc(Cl)c(Cl)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
50
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602165
(CHEMBL5193084)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
63
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571638
(CHEMBL4845759)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1ccc2cnsc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
85
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571571
(CHEMBL4849726)
Show SMILES
Clc1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
89
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571619
(CHEMBL4873593)
Show SMILES
Fc1cc2sncc2cc1NCc1ncc(Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
98
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602162
(CHEMBL5194924)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
100
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571639
(CHEMBL4862183)
Show SMILES
Cn1c(Cl)cnc1CNc1cc2sncc2cc1F
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
102
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602168
(CHEMBL5192928)
Show SMILES
OC[C@H]1Cc2cc(ccc2[C@H](N1)c1cc(F)cc(Cl)c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
125
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602168
(CHEMBL5192928)
Show SMILES
OC[C@H]1Cc2cc(ccc2[C@H](N1)c1cc(F)cc(Cl)c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
126
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571605
(CHEMBL4869736)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
158
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571607
(CHEMBL4863223)
Show SMILES
Cn1c(Cl)cnc1CN(CC1CC1)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
158
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602164
(CHEMBL5186500)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(F)cc(F)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
200
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602163
(CHEMBL5189636)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cc(Cl)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
200
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602170
(CHEMBL5188072)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1cc(F)cc(c1)C#N |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
251
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571640
(CHEMBL4866122)
Show SMILES
Cn1c(Cl)cnc1CNc1ccc2cnsc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
295
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571641
(CHEMBL4849376)
Show SMILES
CN(Cc1ncc(Cl)n1C)c1cc2sncc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
309
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602148
(CHEMBL5181952)
Show SMILES
OC[C@@H]1Cc2cc(Cl)c(F)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
316
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602160
(CHEMBL5179994)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cccc(F)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
316
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571570
(CHEMBL4876211)
Show SMILES
Cn1c(Cl)cnc1CNc1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
331
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571606
(CHEMBL4863555)
Show SMILES
CN(Cc1ncc(Cl)s1)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
447
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571592
(CHEMBL4855887)
Show SMILES
Cn1c(Br)cnc1CNc1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
457
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571611
(CHEMBL4849797)
Show SMILES
CCN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
468
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571620
(CHEMBL4858854)
Show SMILES
Clc1cnc(CNc2cc3cnsc3cn2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
468
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571598
(CHEMBL4874619)
Show SMILES
FC(F)(F)c1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
490
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602159
(CHEMBL5202815)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1cccc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
501
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602147
(CHEMBL5209164)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
501
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571599
(CHEMBL4866780)
Show SMILES
Cc1cnc(CNc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
575
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602135
(CHEMBL5209032)
Show SMILES
Cn1c2ccccc2s\c1=N\C(=S)NCC=C
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
631
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602141
(CHEMBL5175850)
Show SMILES
OC[C@@H]1Cc2ccc(Cl)cc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
794
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571616
(CHEMBL4867011)
Show SMILES
Clc1cnc(COc2ccc3sncc3c2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
832
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571623
(CHEMBL4872165)
Show SMILES
Fc1c(NCc2ncc(Cl)s2)ccc2sncc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
933
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602161
(CHEMBL5184410)
Show SMILES
Cc1cc(ccc1Cl)[C@@H]1N[C@H](CO)Cc2ccc(Cl)cc12 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.00E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571624
(CHEMBL4848175)
Show SMILES
Clc1cnc(CNc2ccc3sncc3n2)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.18E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602149
(CHEMBL5175871)
Show SMILES
OC[C@@H]1Cc2c(Cl)cccc2[C@@H](N1)c1ccccc1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.26E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571627
(CHEMBL4855018)
Show SMILES
Fc1cc(NCc2ncc(Cl)s2)cc2cnsc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.38E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571633
(CHEMBL4871607)
Show SMILES
Clc1cnc(CNc2cccc3cnsc23)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.45E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571622
(CHEMBL4861157)
Show SMILES
Clc1cnc(CNc2ccc3sncc3c2Cl)s1
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.59E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602158
(CHEMBL5169709)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ccc2[C@@H](N1)c1ccccc1Cl |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.59E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571629
(CHEMBL4850037)
Show SMILES
CN(Cc1ncc(Cl)s1)c1cc2cnsc2cc1Cl
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.62E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50571621
(CHEMBL4864644)
Show SMILES
Cc1c(NCc2ncc(Cl)s2)ccc2sncc12
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
1.74E+3
n/a
n/a
n/a
n/a
TBA
Assay Description
Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay
Citation and Details
Article DOI:
10.1021/acs.jmedchem.1c00065
BindingDB Entry DOI:
10.7270/Q2J106ZZ
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5
(Homo sapiens (Human))
BDBM50602166
(CHEMBL5203756)
Show SMILES
OC[C@@H]1Cc2cc(Cl)ncc2[C@@H](N1)c1cc(F)cc(Cl)c1 |r|
Show InChI
UniProtKB/SwissProt
GoogleScholar
AffyNet
PC cid
PC sid
UniChem
Article
PubMed
n/a
n/a
n/a
n/a
2.00E+3
n/a
n/a
n/a
n/a
TBA
Citation and Details
Article DOI:
10.1016/j.bmc.2022.117084
BindingDB Entry DOI:
10.7270/Q2XW4PWD
More data for this
Ligand-Target Pair
Displayed 1 to 50 (of 114 total ) |
Next
|
Last
>>
Jump to: