Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170371 (5-Piperidin-1-ylmethyl-thiazole-4-carboxylic acid ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170370 (5-[2-Methoxy-2-(4-methoxy-phenyl)-ethyl]-thiazole-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169672 (5-(Cyclopentanecarbonyl-amino)-thiazole-4-carboxyl...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170365 (5-Pyrrolidin-1-ylmethyl-thiazole-4-carboxylic acid...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170369 (5-(2-Ethoxy-3-methyl-butyl)-thiazole-4-carboxylic ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169661 (5-(2-Benzyloxy-acetylamino)-thiazole-4-carboxylic ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170378 (5-[2-(4-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170386 (CHEMBL366071 | Phenyl-acetic acid 2-[4-(thiazol-2-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170383 (5-[2-(2-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170367 (5-[2-Methoxy-2-(2-methoxy-phenyl)-ethyl]-thiazole-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170388 (5-((R)-2-Methoxy-2-phenyl-ethyl)-thiazole-4-carbox...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170358 (5-[2-(3-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169669 (5-(Cyclobutanecarbonyl-amino)-thiazole-4-carboxyli...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170364 (Benzoic acid 2-[4-(thiazol-2-ylcarbamoyl)-thiazol-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169676 (5-(Cyclopropanecarbonyl-amino)-thiazole-4-carboxyl...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170382 (5-(2-Methoxy-2-phenyl-ethyl)-thiazole-4-carboxylic...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Staphylococcus aureus) | BDBM17871 ((1S)-1-[5-(benzylsulfanyl)-4H-1,2,4-triazol-3-yl]-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 43.7 | n/a | n/a | n/a | n/a | 7.5 | 22 |
Morphochem AG | Assay Description The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c... | J Mol Biol 332: 13-21 (2003) Article DOI: 10.1016/s0022-2836(03)00862-3 BindingDB Entry DOI: 10.7270/Q2C53J49 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169656 (5-(2-Methyl-but-3-enoylamino)-thiazole-4-carboxyli...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170361 (5-(2-Piperidin-1-yl-ethyl)-thiazole-4-carboxylic a...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169665 (5-But-3-enoylamino-thiazole-4-carboxylic acid thia...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 54 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170389 (5-(2-Cyclohexyl-2-methoxy-ethyl)-thiazole-4-carbox...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 54 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170379 (5-Morpholin-4-ylmethyl-thiazole-4-carboxylic acid ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170366 (5-[2-(4-Fluoro-phenyl)-2-methoxy-ethyl]-thiazole-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169660 (CHEMBL176607 | [4-(Thiazol-2-ylcarbamoyl)-thiazol-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170359 (5-(Methoxy-phenyl-methyl)-thiazole-4-carboxylic ac...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169670 (5-Phenethyl-thiazole-4-carboxylic acid thiazol-2-y...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170384 (5-((S)-2-Methoxy-2-phenyl-ethyl)-thiazole-4-carbox...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169685 (CHEMBL360353 | N-[4-(Thiazol-2-ylcarbamoyl)-thiazo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170387 (5-(2-Methoxy-2-methyl-propyl)-thiazole-4-carboxyli...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169664 (5-(2-Methoxy-propyl)-thiazole-4-carboxylic acid th...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169664 (5-(2-Methoxy-propyl)-thiazole-4-carboxylic acid th...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169658 (5-(2-Fluoro-benzoylamino)-thiazole-4-carboxylic ac...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169667 (Acetic acid [4-(thiazol-2-ylcarbamoyl)-thiazol-5-y...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50180755 (2-thiazol-4-yl-1H-imidazo[4,5-b]pyridine | CHEMBL1...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 78 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University Curated by ChEMBL | Assay Description Inhibition of Co2+ loaded MetAP expressed in Escherichia coli | J Med Chem 49: 511-22 (2006) Article DOI: 10.1021/jm050476z BindingDB Entry DOI: 10.7270/Q2N58KXD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169671 (5-Propionylamino-thiazole-4-carboxylic acid thiazo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 81 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169684 (5-(2-Chloro-4-fluoro-benzyl)-thiazole-4-carboxylic...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 82 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169681 (CHEMBL178736 | N-[4-(Thiazol-2-ylcarbamoyl)-thiazo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 88 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169679 (5-(2-Methoxy-3-methyl-butyl)-thiazole-4-carboxylic...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169679 (5-(2-Methoxy-3-methyl-butyl)-thiazole-4-carboxylic...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170360 (5-(2-Methoxy-4-methyl-pentyl)-thiazole-4-carboxyli...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170374 (5-[2-(3-Chloro-phenyl)-2-methoxy-ethyl]-thiazole-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170376 (5-(2-Benzyloxy-ethyl)-thiazole-4-carboxylic acid t...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169677 (5-(2-Methoxy-acetylamino)-thiazole-4-carboxylic ac...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 92 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170373 (5-Methoxymethyl-thiazole-4-carboxylic acid thiazol...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169683 (5-Isobutyl-thiazole-4-carboxylic acid thiazol-2-yl...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50170381 (5-(2-Methoxy-hexyl)-thiazole-4-carboxylic acid thi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50180731 (2-(pyridin-2-yl)-1H-imidazo[4,5-b]pyridine | 2-pyr...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a | n/a |
Saarland University Curated by ChEMBL | Assay Description Inhibition of Co2+ loaded MetAP expressed in Escherichia coli | J Med Chem 49: 511-22 (2006) Article DOI: 10.1021/jm050476z BindingDB Entry DOI: 10.7270/Q2N58KXD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169662 (CHEMBL175540 | Thiazole-4-carboxylic acid thiazol-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169686 (5-(4-Fluoro-benzoylamino)-thiazole-4-carboxylic ac...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration required against Escherichia coli MetAP1 (150 nM) | Bioorg Med Chem Lett 15: 3732-6 (2005) Article DOI: 10.1016/j.bmcl.2005.05.055 BindingDB Entry DOI: 10.7270/Q2T1534B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Methionine aminopeptidase (Escherichia coli (strain K12)) | BDBM50169662 (CHEMBL175540 | Thiazole-4-carboxylic acid thiazol-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Graduate School of the Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibitory concentration against EcMetAP1 enzyme activity | Bioorg Med Chem Lett 15: 4130-5 (2005) Article DOI: 10.1016/j.bmcl.2005.06.005 BindingDB Entry DOI: 10.7270/Q2FN15RH | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 411 total ) | Next | Last >> |