Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420157 ((7S)-4-[(6-Chloropyrazolo[1,5-a]pyridin-5-yl)amino...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420278 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420249 ((7S)—N-Butyl-4-[(6-methoxypyrazolo[1,5-a]pyridin-5...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420250 (1-((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420251 ((7S)—N-[3-(Dimethylamino)propyl]-4-[(6-methoxypyra...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420252 ((3-Hydroxy-3-methylazetidin-1-yl)(7S)-4-[(6-methox...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420256 ((7S)—N-(2-Methoxyethyl)-4-[(6-methoxypyrazolo[1,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420258 (US10487092, Example 106 | [(3R)-3-(Dimethylamino)p...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420259 (US10487092, Example 107 | [(3S)-3-(Dimethylamino)p...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420260 (US10487092, Example 108 | [(3S,4S)-3,4-Dihydroxypy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420261 (US10487092, Example 109 | [4-(Dimethylamino)piperi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420262 ((4-[2-Dimethylamino)ethyl]methyl)aminopiperidin-1-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420265 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420266 (4-[2-(Dimethylamino)ethyl]piperazin-1-yl(7S)-4-[(6...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420267 ((7S)—N-[2-(Dimethylamino)ethyl]-N-ethyl-4-[(6-meth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420268 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420269 ((7S)—N-Ethyl-N-(2-hydroxyethyl)-4-[(6-methoxypyraz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420270 ((7S)—N-Ethyl-N-(2-methoxyethyl)-4-[(6-methoxypyraz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420271 ((7S)—N,N-Bis(2-methoxyethyl)-4-[(6-methoxypyrazolo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420273 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420274 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420276 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420277 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420246 ((7S)—N-Ethyl-4-[(6-methoxypyrazolo[1,5-a]pyridin-5...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM223024 (US9320737, II.1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 7.5 | 22 |
BAYER INTELLECTUAL PROPERTY GMBH US Patent | Assay Description For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9320737 (2016) BindingDB Entry DOI: 10.7270/Q22V2F00 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM223030 (US9320737, III.3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 7.5 | 22 |
BAYER INTELLECTUAL PROPERTY GMBH US Patent | Assay Description For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9320737 (2016) BindingDB Entry DOI: 10.7270/Q22V2F00 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM223043 (US9320737, IV.2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 7.5 | 22 |
BAYER INTELLECTUAL PROPERTY GMBH US Patent | Assay Description For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9320737 (2016) BindingDB Entry DOI: 10.7270/Q22V2F00 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420155 ((7S)-4-[(6-Chloropyrazolo[1,5-a]pyridin-5-yl)amino...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420195 ((7S)—N-(2-Hydroxy-2-methylpropyl)-4-[(6-methoxypyr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420275 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420253 ((7S)—N-[2-(Dimethylamino)ethyl]-4-[(6-methoxypyraz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420254 (US10487092, Example 102 | [3-(Dimethylamino)azetid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420257 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420264 (US10487092, Example 112 | [(2R,6S)-2,6-Dimethylmor...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420247 ((7S)—N-(2,2-Difluoroethyl)-4-[(6-methoxypyrazolo[1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337234 (N-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420263 ((7S)—N-[3-(Dimethylamino)propyl]-N-(2-hydroxyethyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337242 ((5S)-1-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridaz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337246 ((2R)-2-hydroxy-N-[3-(4-methoxyfuro[3,2-c]pyridin-2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337234 (N-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337240 (N-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337242 ((5S)-1-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridaz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM337246 ((2R)-2-hydroxy-N-[3-(4-methoxyfuro[3,2-c]pyridin-2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (... | US Patent US9745304 (2017) BindingDB Entry DOI: 10.7270/Q2D79DHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420193 ((7S)—N-(2,2-Difluoroethyl)-4-[(6-methoxypyrazolo[1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420194 ((7S)-4-[(6-Methoxypyrazolo[1,5-a]pyridin-5-yl)amin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420196 ((7S)—N-[2-(Dimethylamino)ethyl]-4-[(6-methoxypyraz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420197 ((7S)—N-(2-Hydroxyethyl)-4-[(6-methoxypyrazolo[1,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420198 ((7S)—N-(2-Methoxyethyl)-4-[(6-methoxypyrazolo[1,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420222 ((7S)—N-(1H-Indol-5-yl)-4-[(6-methoxypyrazolo[1,5-a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D] (Homo sapiens (Human)) | BDBM420255 ((7S)—N-(2-Hydroxyethyl)-4-[(6-methoxypyrazolo [1,5...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
BAYER PHARMA AKTIENGESELLSCHAFT US Patent | Assay Description A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n... | US Patent US10487092 (2019) BindingDB Entry DOI: 10.7270/Q28W3GPZ | |||||||||||
More data for this Ligand-Target Pair |
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