Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50035297 (CHEBI:28862 | CHEMBL1232205) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM92459 (CHEMBL384759 | GDP | Guanosine Diphosphate) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 5.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50370754 (CHEMBL252929) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50035296 (CHEMBL3343356) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.04E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50035294 (CHEMBL3343358) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.34E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50035295 (CHEMBL3343357) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.39E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 (Homo sapiens (Human)) | BDBM50035293 (CHEMBL3343359) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.47E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hamburg University Curated by ChEMBL | Assay Description Inhibition of human recombinant alpha1,3-fucosyltransferase 9 using GDP-[14C]-fucose preincubated for 30 mins by liquid scintillation counting | Bioorg Med Chem 22: 6430-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.038 BindingDB Entry DOI: 10.7270/Q2G73GC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1,3-galactosyltransferase 1 (Homo sapiens (Human)) | BDBM50427122 (CHEMBL2323431) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University Curated by ChEMBL | Assay Description Inhibition of human recombinant soluble His-tagged beta3-GalT1 expressed in insect cells using GlcNAcbeta-Bn as substrate after 1 hr | Bioorg Med Chem 21: 1305-11 (2013) Article DOI: 10.1016/j.bmc.2012.12.034 BindingDB Entry DOI: 10.7270/Q2J67J72 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1,3-galactosyltransferase 1 (Homo sapiens (Human)) | BDBM50427121 (CHEMBL2323429 | CHEMBL2323430) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University Curated by ChEMBL | Assay Description Inhibition of human recombinant soluble His-tagged beta3-GalT1 expressed in insect cells using GlcNAcbeta-Bn as substrate after 1 hr | Bioorg Med Chem 21: 1305-11 (2013) Article DOI: 10.1016/j.bmc.2012.12.034 BindingDB Entry DOI: 10.7270/Q2J67J72 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1,3-galactosyltransferase 1 (Homo sapiens (Human)) | BDBM50427121 (CHEMBL2323429 | CHEMBL2323430) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University Curated by ChEMBL | Assay Description Inhibition of human recombinant soluble His-tagged beta3-GalT1 expressed in insect cells using GlcNAcbeta-Bn as substrate after 1 hr | Bioorg Med Chem 21: 1305-11 (2013) Article DOI: 10.1016/j.bmc.2012.12.034 BindingDB Entry DOI: 10.7270/Q2J67J72 | |||||||||||
More data for this Ligand-Target Pair |