Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020375 (CHEMBL3289785) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50499936 (CHEMBL3742171) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Toyama Prefectural University Curated by ChEMBL | Assay Description Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysis | J Nat Prod 78: 2827-31 (2015) Article DOI: 10.1021/acs.jnatprod.5b00540 BindingDB Entry DOI: 10.7270/Q20868BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50499937 (CHEBI:67522 | Turnagainolide A) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Toyama Prefectural University Curated by ChEMBL | Assay Description Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysis | J Nat Prod 78: 2827-31 (2015) Article DOI: 10.1021/acs.jnatprod.5b00540 BindingDB Entry DOI: 10.7270/Q20868BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50499939 (CHEMBL3740058) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Toyama Prefectural University Curated by ChEMBL | Assay Description Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysis | J Nat Prod 78: 2827-31 (2015) Article DOI: 10.1021/acs.jnatprod.5b00540 BindingDB Entry DOI: 10.7270/Q20868BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50499938 (CHEMBL3741390) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Toyama Prefectural University Curated by ChEMBL | Assay Description Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysis | J Nat Prod 78: 2827-31 (2015) Article DOI: 10.1021/acs.jnatprod.5b00540 BindingDB Entry DOI: 10.7270/Q20868BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50351512 (CHEMBL8483) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Nottingham Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus RN6390B Agr-mediated RNA3 promoter activation measured up to 6 hrs by Northern blot analysis | J Med Chem 56: 1389-404 (2013) Article DOI: 10.1021/jm3014635 BindingDB Entry DOI: 10.7270/Q2BV7J0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020376 (CHEBI:81348 | CHEMBL290932) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020377 (CHEMBL3289786) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM11318 (1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.71E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020378 (CHEMBL3289787) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020379 (CHEMBL3289788) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020380 (CHEMBL3289789) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM115127 (4,5,7-trihydroxy-9,10-diketo-anthracene-2-carboxyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.06E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50312649 (6-chloro-4,5,7-trihydroxy-9,10-dioxo-9,10-dihydroa...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.78E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Accessory gene regulator protein A (Staphylococcus aureus) | BDBM50020389 (CHEMBL3289790) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Greensboro Curated by ChEMBL | Assay Description Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assay | J Nat Prod 77: 1351-8 (2014) Article DOI: 10.1021/np5000704 BindingDB Entry DOI: 10.7270/Q21V5GJD | |||||||||||
More data for this Ligand-Target Pair |