Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytochrome P450 26B1 (Homo sapiens (Human)) | BDBM50253810 (CHEMBL459505 | N-(4-(2-ethyl-1-(1H-1,2,4-triazol-1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington at Seattle | Assay Description Eighteen compounds were tested as potential inhibitors of CYP26A1 and CYP26B1. The formation of 9-cis-4-OH-RA metabolite was monitored and the percen... | J Med Chem 52: 1864-72 (2009) BindingDB Entry DOI: 10.7270/Q2FN18J2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 26B1 (Homo sapiens (Human)) | BDBM50253810 (CHEMBL459505 | N-(4-(2-ethyl-1-(1H-1,2,4-triazol-1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Inhibition of microsomal fraction of human CYP26B1 expressed in Sf9 cells using 9-cis-RA as substrate preincubated for 5 mins followed by NADPH addit... | J Med Chem 59: 2579-95 (2016) Article DOI: 10.1021/acs.jmedchem.5b01780 BindingDB Entry DOI: 10.7270/Q2J38VG8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558426 (Methyl 4-hydroxy-4-[3-[[6-(1-H-pyrazol-5-yl)-3-pyr...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558265 (N-Methyl-3-[[methyl-[3-[[6-(1-H-pyrazol-5-yl)-3-py...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 26B1 (Homo sapiens (Human)) | BDBM393281 (US9963439, R116010) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington at Seattle | Assay Description Eighteen compounds were tested as potential inhibitors of CYP26A1 and CYP26B1. The formation of 9-cis-4-OH-RA metabolite was monitored and the percen... | J Med Chem 52: 1864-72 (2009) BindingDB Entry DOI: 10.7270/Q2FN18J2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558427 (US11365192, Example 51-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558428 (1-[4-Hydroxy-4-[3-[[6-(1-H-pyrazol-5-yl)-3-pyridin...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558214 (2,3-Difluoro-5-[3-[[6-(1H-pyrazol-5-yl)-3-pyridiny...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558439 (N-Methyl-N-[[3-[[6-(1H-pyrazol-5-yl)-3-pyridinyl]o...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558338 (US11365192, Example 42-16) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558218 (2-Methyl-5-[[6-(1H-pyrazol-5-yl)-3-pyridinyl]oxyme...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558269 (US11365192, Example 23-6) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM50591500 (CHEMBL5195099) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01089 BindingDB Entry DOI: 10.7270/Q2MK6HW6 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558216 (US11365192, Example 11-3) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558188 (1-Acetyl-4-[8-[[6-(1H-pyrazol-5-yl)-3-pyridinyl]ox...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558158 (US11365192, Example 1-63) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558529 (US11365192, Example 72-6) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558440 (1,1,1-Trifluoro-3-[3-[[6-(1H-pyrazol-5-yl)-3-pyrid...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558342 (US11365192, Example 42-20) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558219 (US11365192, Example 12-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558326 (US11365192, Example 42-4) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558533 (1,1-Dioxo-3-[8-[6-(1H-pyrazol-5-yl)pyridin-3-yl]ox...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558339 (US11365192, Example 42-17) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558222 (US11365192, Example 13-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558527 (US11365192, Example 72-4) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558335 (US11365192, Example 42-13) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM50591501 (CHEMBL5183418) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01089 BindingDB Entry DOI: 10.7270/Q2MK6HW6 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558332 (US11365192, Example 42-10) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558431 (US11365192, Example 53-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558452 (3-[[6-(4-Chloro-1H-pyrazol-5-yl)-3-pyridinyl]oxyme...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM50591496 (CHEMBL5204432) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01089 BindingDB Entry DOI: 10.7270/Q2MK6HW6 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 26B1 (Homo sapiens (Human)) | BDBM50157605 (Liarozole | Liazal | R-75251 | US9963439, Liarozol...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington at Seattle | Assay Description Eighteen compounds were tested as potential inhibitors of CYP26A1 and CYP26B1. The formation of 9-cis-4-OH-RA metabolite was monitored and the percen... | J Med Chem 52: 1864-72 (2009) BindingDB Entry DOI: 10.7270/Q2FN18J2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 26B1 (Homo sapiens (Human)) | BDBM50157605 (Liarozole | Liazal | R-75251 | US9963439, Liarozol...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Inhibition of microsomal fraction of human CYP26B1 expressed in Sf9 cells using 9-cis-RA as substrate preincubated for 5 mins followed by NADPH addit... | J Med Chem 59: 2579-95 (2016) Article DOI: 10.1021/acs.jmedchem.5b01780 BindingDB Entry DOI: 10.7270/Q2J38VG8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558532 (US11365192, Example 72-9) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558360 (US11365192, Example 43-14) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558215 (US11365192, Example 11-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558140 (US11365192, Example 1-45) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM50591519 (CHEMBL5174407) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01089 BindingDB Entry DOI: 10.7270/Q2MK6HW6 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558223 (US11365192, Example 13-3) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558552 (US11365192, Example 75-7 | US11365192, Example 75-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558359 (US11365192, Example 43-13) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558340 (US11365192, Example 42-18) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM50591499 (CHEMBL5173608) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01089 BindingDB Entry DOI: 10.7270/Q2MK6HW6 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558236 (N-[6-[[6-(1H-Pyrazol-5-yl)-3-pyridinyl]oxy]hexyl]m...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558362 (US11365192, Example 43-16) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558173 (4-[8-[[6-(1H-Pyrazol-5-yl)-3-pyridinyl]oxy]octyl]-...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558324 (US11365192, Example 42-2) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558220 (US11365192, Example 12-3) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558467 (US11365192, Example 70-5) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 4F2 (Homo sapiens (Human)) | BDBM558343 (US11365192, Example 42-21) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In the CYP4F2 inhibition test, the reaction solution containing each compound [final concentration of 50 mM, KPO4 (pH 7.4), 2.5 μM luciferine de... | Citation and Details BindingDB Entry DOI: 10.7270/Q2PN98V9 | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 572 total ) | Next | Last >> |