Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106707 (CHEMBL1957358 | US8586620, 67) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106699 (CHEMBL1957350 | US8586620, 46) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106698 (CHEMBL1957349 | US8586620, 42) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106706 (CHEMBL1957356 | US8586620, 64) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM50005835 ((3-[2-(dimethylamino)ethyl]-1H-indol-5-yl)-N-methy...) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents | US Patent | n/a | n/a | 59 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106715 (US8586620, 97) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106701 (CHEMBL1957352 | US8586620, 51) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106700 (CHEMBL1957354 | US8586620, 47) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106704 (US8586620, 59) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106720 (US8586620, 110) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106696 (US8586620, 56) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106721 (US8586620, 111) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106697 (CHEMBL1957353 | US8586620, 43) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106705 (US8586620, 62) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106703 (US8586620, 15) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 870 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine 1D receptor (Bos taurus (Bovine)) | BDBM106717 (US8586620, 105) | PDB Reactome pathway UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
NeurAxon, Inc. US Patent | Assay Description 5-HT1D binding assays (agonist radioligand)were performed using bovine caudate membranes according to the methods of Heuring and Peroutka (J. Neurosc... | US Patent US8586620 (2013) BindingDB Entry DOI: 10.7270/Q2348J0K | |||||||||||
More data for this Ligand-Target Pair |