Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1 (Homo sapiens (Human)) | BDBM50004840 (Amino-(4-phosphonomethyl-phenyl)-acetic acid | CHE...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a |
Novartis Pharma AG Curated by ChEMBL | Assay Description Dissociation constant of the compound against N-methyl-D-aspartate glutamate receptor using [3H]-CPP binding was determined | Bioorg Med Chem Lett 10: 1241-4 (2000) BindingDB Entry DOI: 10.7270/Q26972SC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50414372 (CHEMBL2145458) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a |
University of Berne Curated by ChEMBL | Assay Description Activity at rat NR1/NR2A receptor expressed in Xenopus oocytes assessed as inhibition of glycine-induced electrophysiological response | Bioorg Med Chem Lett 19: 3832-5 (2009) Article DOI: 10.1016/j.bmcl.2009.04.021 BindingDB Entry DOI: 10.7270/Q2Z0386F | |||||||||||
More data for this Ligand-Target Pair |