Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254202 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-3-(2-amino-2-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3beta1 expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair |