Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50037557 (2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human NPFFR1 expressed in green monkey COS-7 cell membranes by [125I]-1DMeNPFF radioligand based saturation binding assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00643 BindingDB Entry DOI: 10.7270/Q2SJ1QC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50060728 ((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 20.9 | n/a | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50394976 (CHEMBL2165922) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 41.7 | n/a | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair |