Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histo-blood group ABO system transferase (Homo sapiens (Human)) | BDBM50427444 (CHEMBL2326313) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.82E+5 | n/a | n/a | n/a | n/a | n/a |
University of Hamburg Curated by ChEMBL | Assay Description Binding affinity to human blood group B Galactosyltransferase by STD NMR analysis in presence of magnesium ions | J Med Chem 56: 2150-4 (2013) Article DOI: 10.1021/jm300642a BindingDB Entry DOI: 10.7270/Q26T0P01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histo-blood group ABO system transferase (Homo sapiens (Human)) | BDBM50427444 (CHEMBL2326313) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.54E+5 | n/a | n/a | n/a | n/a | n/a |
University of Hamburg Curated by ChEMBL | Assay Description Binding affinity to human blood group B Galactosyltransferase after 300 secs by SPR analysis | J Med Chem 56: 2150-4 (2013) Article DOI: 10.1021/jm300642a BindingDB Entry DOI: 10.7270/Q26T0P01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histo-blood group ABO system transferase (Homo sapiens (Human)) | BDBM50427445 (CHEMBL1235497) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.30E+6 | n/a | n/a | n/a | n/a | n/a |
University of Hamburg Curated by ChEMBL | Assay Description Binding affinity to human blood group B Galactosyltransferase after 300 secs by SPR analysis | J Med Chem 56: 2150-4 (2013) Article DOI: 10.1021/jm300642a BindingDB Entry DOI: 10.7270/Q26T0P01 | |||||||||||
More data for this Ligand-Target Pair |