Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bifunctional protein GlmU (Staphylococcus aureus) | BDBM50365075 (CHEMBL1951164 | Sulfonamide, 2) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.30E+3 | 1.90E+3 | n/a | n/a | n/a | 7.35 | n/a |
AstraZeneca | Assay Description Inhibition assay using GlmU bifuncation enzyme with various bacterial strains. | J Biol Chem 286: 40734-42 (2011) Article DOI: 10.1074/jbc.M111.274068 BindingDB Entry DOI: 10.7270/Q2BP01DD | |||||||||||
More data for this Ligand-Target Pair |