Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92704 (Photoaffinity ligand, 1) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 0.440 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92706 (Photoaffinity ligand, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 0.490 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92707 (Photoaffinity ligand, 4) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 0.760 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92705 (Photoaffinity ligand, 2) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 2.10 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM50506039 (CHEMBL1324296) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a |
University of Perugia Curated by ChEMBL | Assay Description Displacement of [3H]TCDD from mouse AhR | Eur J Med Chem 185: (2020) Article DOI: 10.1016/j.ejmech.2019.111842 BindingDB Entry DOI: 10.7270/Q2N019SX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92709 (Photoaffinity ligand, 6) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 8.10 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92711 (Photoaffinity ligand, 8) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 11 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92708 (Photoaffinity ligand, 5) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | 13 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM50239186 (1,1-Bis(3''-Indolyl)Methane | 3,3''-Diindolylmetha...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a |
University of Perugia Curated by ChEMBL | Assay Description Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR | Eur J Med Chem 185: (2020) Article DOI: 10.1016/j.ejmech.2019.111842 BindingDB Entry DOI: 10.7270/Q2N019SX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Mus musculus (Mouse)) | BDBM92710 (Photoaffinity ligand, 7) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 113 | n/a | n/a | n/a | 7.5 | 0 |
University of Wisconsin | Assay Description The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. | J Biol Chem 261: 6352-65 (1986) BindingDB Entry DOI: 10.7270/Q2X928X8 | |||||||||||
More data for this Ligand-Target Pair |