Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM50020938 (CHEMBL3287301) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Binding affinity to Bcl-w (unknown origin) by surface plasmon resonance assay | ACS Med Chem Lett 5: 662-7 (2014) Article DOI: 10.1021/ml500030p BindingDB Entry DOI: 10.7270/Q2KP83QG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM21400 (CHEMBL192571 | N-[(4-{[(2R)-4-(dimethylamino)-1-(p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 459 | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description Binding affinity to Bclw | J Med Chem 49: 1165-81 (2006) Article DOI: 10.1021/jm050754u BindingDB Entry DOI: 10.7270/Q2VM4BT0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM109236 (WEHI-539) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 4.10E+3 | >550 | n/a | n/a | n/a | 7.4 | n/a |
Walter and Eliza Hall Institute of Medical Research, Parkville, Victoria, Australia | Assay Description The protocols for tight and weak binders were described in Biacore S51 assay set-up with a flow rate of 30 µL/min. For His-Bcl-2 protein assays... | Nat Chem Biol 9: 390-7 (2013) Article DOI: 10.1038/nchembio.1246 BindingDB Entry DOI: 10.7270/Q2QJ7FZ7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM50020930 (CHEMBL3287293) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Binding affinity to Bcl-w (unknown origin) by surface plasmon resonance assay | ACS Med Chem Lett 5: 662-7 (2014) Article DOI: 10.1021/ml500030p BindingDB Entry DOI: 10.7270/Q2KP83QG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM50576622 (CHEMBL4850731) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human partial length BCLW (M1 to R171 residues) expressed in bacterial expression system by BCL2SCAN assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00682 BindingDB Entry DOI: 10.7270/Q2MC93VV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 2 (Homo sapiens (Human)) | BDBM50020929 (CHEMBL3287292) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a |
Genentech Curated by ChEMBL | Assay Description Binding affinity to Bcl-w (unknown origin) by surface plasmon resonance assay | ACS Med Chem Lett 5: 662-7 (2014) Article DOI: 10.1021/ml500030p BindingDB Entry DOI: 10.7270/Q2KP83QG | |||||||||||
More data for this Ligand-Target Pair |