Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097567 (CHEMBL3588871) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 240 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097570 (CHEMBL3590074) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097565 (CHEMBL3589947) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097560 (CHEMBL3590072) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097564 (CHEMBL3589948) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097569 (CHEMBL3590075) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097568 (CHEMBL3590076) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097563 (CHEMBL3590069) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097559 (CHEMBL3590073) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097562 (CHEMBL3590070) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097561 (CHEMBL3590071) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50097566 (CHEMBL3589946) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay | Bioorg Med Chem 23: 3913-24 (2015) Article DOI: 10.1016/j.bmc.2014.12.007 BindingDB Entry DOI: 10.7270/Q2MS3VHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50071956 (CHEMBL3407845) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a |
Sorbonne Universit£s Curated by ChEMBL | Assay Description Induction of calcium release in mouse FPR2 receptor-expressed HEK cell by cytosolic-free calcium assay | J Med Chem 58: 1089-99 (2015) Article DOI: 10.1021/jm501018q BindingDB Entry DOI: 10.7270/Q2CN75KX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor-related sequence 1 (Mus musculus) | BDBM50050937 ((S)-2-[(S)-2-((S)-2-Formylamino-4-methylsulfanyl-b...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | >300 | n/a | n/a | n/a | n/a | n/a |
Sorbonne Universit£s Curated by ChEMBL | Assay Description Binding affinity to mouse FPR2 receptor | J Med Chem 58: 1089-99 (2015) Article DOI: 10.1021/jm501018q BindingDB Entry DOI: 10.7270/Q2CN75KX | |||||||||||
More data for this Ligand-Target Pair |