Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ABC-type glutathione-S-conjugate transporter (Homo sapiens (Human)) | BDBM50391002 (CHEMBL2074599) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | PubMed | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cells | Pharm Res 19: 34-41 (2002) BindingDB Entry DOI: 10.7270/Q2G44RCW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ABC-type glutathione-S-conjugate transporter (Homo sapiens (Human)) | BDBM50391003 (CHEMBL493586) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | PubMed | 1.05E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cells | Pharm Res 19: 34-41 (2002) BindingDB Entry DOI: 10.7270/Q2G44RCW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ABC-type glutathione-S-conjugate transporter (Homo sapiens (Human)) | BDBM50391004 (CHEMBL213947) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid UniChem Similars | PubMed | 3.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cells | Pharm Res 19: 34-41 (2002) BindingDB Entry DOI: 10.7270/Q2G44RCW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ABC-type glutathione-S-conjugate transporter (Homo sapiens (Human)) | BDBM18050 (2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.20E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cells | Pharm Res 19: 34-41 (2002) BindingDB Entry DOI: 10.7270/Q2G44RCW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ABC-type glutathione-S-conjugate transporter (Homo sapiens (Human)) | BDBM50375594 (TAUROCHOLATE) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.4 uM) in membrane vesicles from MRP3-expressing HEK cells | Biochemistry 42: 9989-10000 (2003) Article DOI: 10.1021/bi034462b BindingDB Entry DOI: 10.7270/Q2JM2BXS | |||||||||||
More data for this Ligand-Target Pair |