Found 427 hits Enz. Inhib. hit(s) with Target = 'Protein delta homolog 1' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50441567
(CHEMBL2436978 | US10485800, Example 181)Show SMILES CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1 Show InChI InChI=1S/C27H27N5/c1-31-10-12-32(13-11-31)18-19-2-4-20(5-3-19)23-15-24-25(17-30-27(24)29-16-23)21-6-7-26-22(14-21)8-9-28-26/h2-9,14-17,28H,10-13,18H2,1H3,(H,29,30) | KEGG
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| n/a | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a |
Califia Bio Inc.
Curated by ChEMBL
| Assay Description
Binding affinity to human wild type DLK by qPCR analysis |
J Med Chem 56: 8032-48 (2013)
Article DOI: 10.1021/jm401094t
BindingDB Entry DOI: 10.7270/Q2P270KS |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM4814
(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)Show SMILES CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C Show InChI InChI=1S/C22H27FN4O2/c1-5-27(6-2)10-9-24-22(29)20-13(3)19(25-14(20)4)12-17-16-11-15(23)7-8-18(16)26-21(17)28/h7-8,11-12,25H,5-6,9-10H2,1-4H3,(H,24,29)(H,26,28)/b17-12- | KEGG
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| n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50308060
(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)Show SMILES C[C@]12O[C@H](C[C@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13 |r| Show InChI InChI=1S/C26H21N3O4/c1-25-26(32,12-30)10-18(33-25)28-16-8-4-2-6-13(16)20-21-15(11-27-24(21)31)19-14-7-3-5-9-17(14)29(25)23(19)22(20)28/h2-9,18,30,32H,10-12H2,1H3,(H,27,31)/t18-,25+,26+/m1/s1 | KEGG
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| n/a | n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50326053
(CHEMBL608533 | PKC-412)Show SMILES CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r| Show InChI InChI=1S/C35H30N4O4/c1-35-32(42-3)25(37(2)34(41)19-11-5-4-6-12-19)17-26(43-35)38-23-15-9-7-13-20(23)28-29-22(18-36-33(29)40)27-21-14-8-10-16-24(21)39(35)31(27)30(28)38/h4-16,25-26,32H,17-18H2,1-3H3,(H,36,40)/t25-,26-,32-,35+/m1/s1 | KEGG
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| n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50300690
(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)Show SMILES CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1 Show InChI InChI=1S/C29H32N6O4S/c1-29(2,3)25-17-26(33-39-25)32-27(36)30-20-6-4-19(5-7-20)22-18-35-23-9-8-21(16-24(23)40-28(35)31-22)38-15-12-34-10-13-37-14-11-34/h4-9,16-18H,10-15H2,1-3H3,(H2,30,32,33,36) | KEGG
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| n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM16673
(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)Show SMILES CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1 Show InChI InChI=1S/C21H16ClF3N4O3/c1-26-19(30)18-11-15(8-9-27-18)32-14-5-2-12(3-6-14)28-20(31)29-13-4-7-17(22)16(10-13)21(23,24)25/h2-11H,1H3,(H,26,30)(H2,28,29,31) | KEGG
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| n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM13535
(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)Show SMILES COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1 Show InChI InChI=1S/C31H42N6O4/c1-23(2)41-25-10-8-24(9-11-25)34-31(38)37-17-15-36(16-18-37)30-26-20-28(39-3)29(21-27(26)32-22-33-30)40-19-7-14-35-12-5-4-6-13-35/h8-11,20-23H,4-7,12-19H2,1-3H3,(H,34,38) | KEGG
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Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50326054
(CHEMBL1240703)Show SMILES CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r| Show InChI InChI=1S/C35H30N4O5/c1-35-31(43-3)23(37(2)34(42)18-11-5-4-6-12-18)17-24(44-35)38-21-15-9-7-13-19(21)25-27-28(33(41)36-32(27)40)26-20-14-8-10-16-22(20)39(35)30(26)29(25)38/h4-16,23-24,31,33,41H,17H2,1-3H3,(H,36,40)/t23-,24-,31-,33+,35+/m1/s1 | KEGG
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| n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
Ambit Biosciences
Curated by ChEMBL
| Assay Description
Binding affinity to DLK |
Blood 114: 2984-92 (2009)
Article DOI: 10.1182/blood-2009-05-222034
BindingDB Entry DOI: 10.7270/Q2PN95V2 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50042942
(CHEMBL3355003)Show SMILES CC(C)n1nc(cc1C1CCN(C)CC1)-c1cnc2[nH]cc(c2c1)C(F)(F)F Show InChI InChI=1S/C20H24F3N5/c1-12(2)28-18(13-4-6-27(3)7-5-13)9-17(26-28)14-8-15-16(20(21,22)23)11-25-19(15)24-10-14/h8-13H,4-7H2,1-3H3,(H,24,25) | KEGG
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| 0.170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) by RT-FRET assay |
ACS Med Chem Lett 6: 11-2 (2015)
Article DOI: 10.1021/ml500347s
BindingDB Entry DOI: 10.7270/Q26W9CQT |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50042940
(CHEMBL3355005)Show SMILES [H][C@@]12CN(C[C@]1([H])[C@H]2c1cc(nn1C(C)C)-c1cnc2[nH]cc(c2c1)C(F)(F)F)C1COC1 |r| | KEGG
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| 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) by RT-FRET assay |
ACS Med Chem Lett 6: 11-2 (2015)
Article DOI: 10.1021/ml500347s
BindingDB Entry DOI: 10.7270/Q26W9CQT |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM4814
(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)Show SMILES CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C Show InChI InChI=1S/C22H27FN4O2/c1-5-27(6-2)10-9-24-22(29)20-13(3)19(25-14(20)4)12-17-16-11-15(23)7-8-18(16)26-21(17)28/h7-8,11-12,25H,5-6,9-10H2,1-4H3,(H,24,29)(H,26,28)/b17-12- | KEGG
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| 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) |
J Med Chem 61: 8078-8087 (2018)
Article DOI: 10.1021/acs.jmedchem.8b00370
BindingDB Entry DOI: 10.7270/Q2G163G3 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50004205
(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)Show SMILES CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1 Show InChI InChI=1S/C23H28N8OS/c1-15-13-20(29-28-15)25-19-14-21(31-11-9-30(2)10-12-31)27-23(26-19)33-18-7-5-17(6-8-18)24-22(32)16-3-4-16/h5-8,13-14,16H,3-4,9-12H2,1-2H3,(H,24,32)(H2,25,26,27,28,29) | KEGG
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| 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) |
J Med Chem 61: 8078-8087 (2018)
Article DOI: 10.1021/acs.jmedchem.8b00370
BindingDB Entry DOI: 10.7270/Q2G163G3 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50042941
(CHEMBL3355004)Show SMILES CC(C)n1nc(cc1C1CCN(C1)C1COC1)-c1cnc2[nH]cc(F)c2c1 | KEGG
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| CHEMBL
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PC sid
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| 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) by RT-FRET assay |
ACS Med Chem Lett 6: 11-2 (2015)
Article DOI: 10.1021/ml500347s
BindingDB Entry DOI: 10.7270/Q26W9CQT |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50042939
(CHEMBL3355006)Show SMILES [H][C@@]12CN(C[C@]1([H])[C@H]2c1cc(nn1C(C)C)-c1cnc(N)c2cn[nH]c12)C1COC1 |r| | KEGG
UniProtKB/SwissProt
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| CHEMBL
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PC sid
UniChem
Similars
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| 270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd.
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) by RT-FRET assay |
ACS Med Chem Lett 6: 11-2 (2015)
Article DOI: 10.1021/ml500347s
BindingDB Entry DOI: 10.7270/Q26W9CQT |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50441567
(CHEMBL2436978 | US10485800, Example 181)Show SMILES CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1 Show InChI InChI=1S/C27H27N5/c1-31-10-12-32(13-11-31)18-19-2-4-20(5-3-19)23-15-24-25(17-30-27(24)29-16-23)21-6-7-26-22(14-21)8-9-28-26/h2-9,14-17,28H,10-13,18H2,1H3,(H,29,30) | KEGG
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| n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Califia Bio Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human wild type DLK by qPCR analysis |
J Med Chem 56: 8032-48 (2013)
Article DOI: 10.1021/jm401094t
BindingDB Entry DOI: 10.7270/Q2P270KS |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50429477
(CHEMBL2332840)Show SMILES FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ncnc4n[nH]cc34)cc2)ccc1Cl Show InChI InChI=1S/C19H12ClF3N6O2/c20-15-6-3-11(7-14(15)19(21,22)23)28-18(30)27-10-1-4-12(5-2-10)31-17-13-8-26-29-16(13)24-9-25-17/h1-9H,(H2,27,28,30)(H,24,25,26,29) | KEGG
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| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sichuan University
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) |
J Med Chem 56: 1641-55 (2013)
Article DOI: 10.1021/jm301537p
BindingDB Entry DOI: 10.7270/Q29S1SC5 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50458548
(CHEMBL4218417)Show SMILES CC(C)OCc1ccc2n(CCO)c3c4[nH]c5ccccc5c4c4CNC(=O)c4c3c2c1 Show InChI InChI=1S/C26H25N3O3/c1-14(2)32-13-15-7-8-20-17(11-15)22-23-18(12-27-26(23)31)21-16-5-3-4-6-19(16)28-24(21)25(22)29(20)9-10-30/h3-8,11,14,28,30H,9-10,12-13H2,1-2H3,(H,27,31) | KEGG
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| n/a | n/a | 119 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]... |
J Med Chem 61: 8078-8087 (2018)
Article DOI: 10.1021/acs.jmedchem.8b00370
BindingDB Entry DOI: 10.7270/Q2G163G3 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM50458549
(CHEMBL4207983)Show SMILES CC(C)n1c2ccc(Oc3ncccn3)cc2c2c3CNC(=O)c3c3-c4cn(C)nc4CCc3c12 Show InChI InChI=1S/C27H24N6O2/c1-14(2)33-21-8-5-15(35-27-28-9-4-10-29-27)11-17(21)23-18-12-30-26(34)24(18)22-16(25(23)33)6-7-20-19(22)13-32(3)31-20/h4-5,8-11,13-14H,6-7,12H2,1-3H3,(H,30,34) | KEGG
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| n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]... |
J Med Chem 61: 8078-8087 (2018)
Article DOI: 10.1021/acs.jmedchem.8b00370
BindingDB Entry DOI: 10.7270/Q2G163G3 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM24942
(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)Show SMILES CCSCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45 |r| Show InChI InChI=1S/C33H33N3O5S2/c1-5-42-15-17-7-9-22-19(11-17)26-27-21(14-34-30(27)37)25-20-12-18(16-43-6-2)8-10-23(20)36-29(25)28(26)35(22)24-13-33(39,31(38)40-4)32(36,3)41-24/h7-12,24,39H,5-6,13-16H2,1-4H3,(H,34,37)/t24-,32+,33+/m1/s1 | KEGG
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| n/a | n/a | 114 | n/a | n/a | n/a | n/a | n/a | n/a |
Genentech
Curated by ChEMBL
| Assay Description
Inhibition of DLK (unknown origin) using myelin basic protein as substrate preincubated for 15 mins measured after 30 mins in presence of [gamma-32P]... |
J Med Chem 61: 8078-8087 (2018)
Article DOI: 10.1021/acs.jmedchem.8b00370
BindingDB Entry DOI: 10.7270/Q2G163G3 |
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637141
(US20230382904, Compound 61)Show SMILES Nc1nc2c(cc(cn2n1)-c1csc(c1)C(=O)NCc1ccc(F)cc1)C(=O)NCC(F)(F)F | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637142
(US20230382904, Compound 62)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NCC(F)(F)F)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637143
(US20230382904, Compound 63)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NCC(F)(F)F)c2nc(N)nn2c1)c1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637144
(US20230382904, Compound 64)Show SMILES Nc1nc2c(cc(cn2n1)-c1csc(c1)C(=O)NCc1ccccc1)C(=O)NC1COC1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637145
(US20230382904, Compound 65)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC2COC2)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637113
(US20230382904, Compound 33 | US20230382904, Compou...)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC2CCNC2)c2nc(N)nn2c1)c1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 88 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637147
(US20230382904, Compound 67)Show SMILES COC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)NCc1ccccc1 |r,$;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;$| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637148
(US20230382904, Compound 68)Show SMILES COC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)NCc1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637149
(US20230382904, Compound 69)Show SMILES COC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637150
(US20230382904, Compound 70)Show SMILES COC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](C)c1ccccc1 |r,$;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;$| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637123
(US20230382904, Compound 43 | US20230382904, Compou...)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)C(F)(F)F)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 4.85 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637123
(US20230382904, Compound 43 | US20230382904, Compou...)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)C(F)(F)F)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637153
(US20230382904, Compound 73)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC2COC2)c2nc(N)nn2c1)c1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637154
(US20230382904, Compound 74)Show SMILES Nc1nc2c(cc(cn2n1)-c1csc(c1)C(=O)NCc1ccc(F)cc1)C(=O)NC1COC1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637155
(US20230382904, Compound 75)Show SMILES CC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC2COC2)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 67 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637156
(US20230382904, Compound 76)Show SMILES CC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)C)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 5.15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637157
(US20230382904, Compound 77)Show SMILES CC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)N[C@@H](C)CO)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637158
(US20230382904, Compound 78)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)(C)CO)c2nc(N)nn2c1)c1ccc(F)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 6.45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637159
(US20230382904, Compound 79)Show SMILES C[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)(C)CO)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637160
(US20230382904, Compound 80)Show SMILES CC(C)(CO)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)NCc1ccc(F)cc1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 56.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637161
(US20230382904, Compound 81)Show SMILES CC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)N[C@@H](C)COC)c2nc(N)nn2c1)c1ccccc1 |r,$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;$| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637162
(US20230382904, Compound 82)Show SMILES CCNC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](CC)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 12.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637163
(US20230382904, Compound 83)Show SMILES CC(C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](C)c1ccc(cc1)C(F)(F)F |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637164
(US20230382904, Compound 84)Show SMILES CC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)(C)C)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637165
(US20230382904, Compound 85)Show SMILES CC(C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(N)=O | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637166
(US20230382904, Compound 86)Show SMILES C[C@@H](CO)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(N)=O |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637167
(US20230382904, Compound 87)Show SMILES CC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)NCc1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637168
(US20230382904, Compound 88)Show SMILES CC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](C)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637169
(US20230382904, Compound 89)Show SMILES CC[C@H](C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](CC)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637170
(US20230382904, Compound 90)Show SMILES CC(C)NC(=O)c1cc(cn2nc(N)nc12)-c1csc(c1)C(=O)N[C@@H](C)c1ccc(C)cc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Protein delta homolog 1
(Homo sapiens (Human)) | BDBM637171
(US20230382904, Compound 91)Show SMILES COC[C@H](NC(=O)c1cc(cs1)-c1cc(C(=O)NC(C)C)c2nc(N)nn2c1)c1ccccc1 |r| | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
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