Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histidine-binding periplasmic protein [1-238] (Escherichia coli (Enterobacteria)) | BDBM7953 ((2S)-2-amino-3-(1H-imidazol-4-yl)propanoic acid | ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 114 | n/a | n/a | n/a | 7.0 | 30 |
University of Calgary | Assay Description All ITC experiments were performed using a Microcal VP-ITC microcalorimeter (GE Healthcare). All samples were prepared in a buffer containing 20 mM H... | J Biol Chem 288: 31409-22 (2013) Article DOI: 10.1074/jbc.M113.490441 BindingDB Entry DOI: 10.7270/Q2862F9B | |||||||||||
More data for this Ligand-Target Pair |