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Found 58 hits Enz. Inhib. hit(s) with Target = 'Lysyl oxidase'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 66n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 83n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 126n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Rattus norvegicus)
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 127n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Mus musculus)
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 128n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Rattus norvegicus)
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 136n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 190n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232681
PNG
(CHEMBL4099444)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 203n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 3


(Homo sapiens (Human))
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 214n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Mus musculus)
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 227n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 243n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232682
PNG
(CHEMBL3467241)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 309n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232693
PNG
(CHEMBL4072524)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 321n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232684
PNG
(CHEMBL4103840)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 385n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 396n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232694
PNG
(CHEMBL4079586)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 431n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase


(Homo sapiens (Human))
BDBM50232678
PNG
(CHEBI:27413 | CHEMBL1618272)
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n/an/a 550n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232691
PNG
(CHEMBL4068773)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 670n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232698
PNG
(CHEMBL1235374)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 719n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232688
PNG
(CHEMBL4075843)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 902n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232685
PNG
(CHEMBL4096085)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 999n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18353
PNG
((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Show SMILES CN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C7H15NO4/c1-8-2-5(10)7(12)6(11)4(8)3-9/h4-7,9-12H,2-3H2,1H3/t4-,5+,6-,7-/m1/s1
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Article
PubMed
n/an/a 1.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18351
PNG
((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Show SMILES OC[C@H]1NC[C@H](O)[C@@H](O)[C@@H]1O
Show InChI InChI=1S/C6H13NO4/c8-2-3-5(10)6(11)4(9)1-7-3/h3-11H,1-2H2/t3-,4+,5-,6-/m1/s1
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PubMed
n/an/a 1.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18366
PNG
((2R,3R,5S,6R)-2,6-bis(hydroxymethyl)piperidine-3,4...)
Show SMILES OC[C@H]1N[C@H](CO)[C@H](O)C(O)[C@@H]1O
Show InChI InChI=1S/C7H15NO5/c9-1-3-5(11)7(13)6(12)4(2-10)8-3/h3-13H,1-2H2/t3-,4-,5-,6+,7?/m1/s1
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n/an/a 1.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232690
PNG
(4-Aminomethyl-Benzamidine | CHEMBL187301)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 1.11E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232683
PNG
(CHEMBL4066086)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 1.18E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232687
PNG
(CHEMBL1188378)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Patents

n/an/a 1.22E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232679
PNG
(CHEMBL4068784)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 1.45E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18358
PNG
((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...)
Show SMILES CCCCCCCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C15H31NO4/c1-2-3-4-5-6-7-8-9-16-10-13(18)15(20)14(19)12(16)11-17/h12-15,17-20H,2-11H2,1H3/t12-,13+,14-,15-/m1/s1
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PubMed
n/an/a 1.50E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18357
PNG
((2R,3R,4R,5S)-2-(hydroxymethyl)-1-octylpiperidine-...)
Show SMILES CCCCCCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C14H29NO4/c1-2-3-4-5-6-7-8-15-9-12(17)14(19)13(18)11(15)10-16/h11-14,16-19H,2-10H2,1H3/t11-,12+,13-,14-/m1/s1
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PubMed
n/an/a 2.10E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232697
PNG
((3-(Methoxycarbonyl)Phenyl)Methanaminium | CHEMBL1...)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 3.54E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50408793
PNG
(CHEMBL148986)
Show SMILES COC(=O)c1ccc(CN)cc1
Show InChI InChI=1S/C9H11NO2/c1-12-9(11)8-4-2-7(6-10)3-5-8/h2-5H,6,10H2,1H3
GoogleScholar
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CHEMBL
PC cid
PC sid
UniChem
n/an/a 3.62E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18356
PNG
((2R,3R,4R,5S)-1-hexyl-2-(hydroxymethyl)piperidine-...)
Show SMILES CCCCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C12H25NO4/c1-2-3-4-5-6-13-7-10(15)12(17)11(16)9(13)8-14/h9-12,14-17H,2-8H2,1H3/t9-,10+,11-,12-/m1/s1
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PubMed
n/an/a 4.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18364
PNG
((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-nonylpiperidi...)
Show SMILES CCCCCCCCC[C@H]1N[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
Show InChI InChI=1S/C15H31NO4/c1-2-3-4-5-6-7-8-9-11-13(18)15(20)14(19)12(10-17)16-11/h11-20H,2-10H2,1H3/t11-,12-,13+,14-,15-/m1/s1
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PubMed
n/an/a 4.80E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232689
PNG
(CHEMBL4098510)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 4.97E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18363
PNG
((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Show SMILES CCCCCCCC[C@H]1N[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
Show InChI InChI=1S/C14H29NO4/c1-2-3-4-5-6-7-8-10-12(17)14(19)13(18)11(9-16)15-10/h10-19H,2-9H2,1H3/t10-,11-,12+,13-,14-/m1/s1
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n/an/a 5.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18355
PNG
((2R,3R,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-...)
Show SMILES CCCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C10H21NO4/c1-2-3-4-11-5-8(13)10(15)9(14)7(11)6-12/h7-10,12-15H,2-6H2,1H3/t7-,8+,9-,10-/m1/s1
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PubMed
n/an/a 5.00E+3n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase


(Homo sapiens (Human))
BDBM50232679
PNG
(CHEMBL4068784)
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n/an/a 5.91E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232695
PNG
(CHEMBL4060123)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 6.04E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232686
PNG
(CHEMBL4088360)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 8.21E+3n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18362
PNG
((2R,3S,4R,5R,6R)-2-hexyl-6-(hydroxymethyl)piperidi...)
Show SMILES CCCCCC[C@H]1N[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
Show InChI InChI=1S/C12H25NO4/c1-2-3-4-5-6-8-10(15)12(17)11(16)9(7-14)13-8/h8-17H,2-7H2,1H3/t8-,9-,10+,11-,12-/m1/s1
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PubMed
n/an/a 1.20E+4n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50113835
PNG
(4-Fluoro-benzylamine | 4-fluorobenzylamine | CHEMB...)
Show SMILES NCc1ccc(F)cc1
Show InChI InChI=1S/C7H8FN/c8-7-3-1-6(5-9)2-4-7/h1-4H,5,9H2
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n/an/a 2.60E+4n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18359
PNG
((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-methylpiperid...)
Show SMILES C[C@H]1N[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
Show InChI InChI=1S/C7H15NO4/c1-3-5(10)7(12)6(11)4(2-9)8-3/h3-12H,2H2,1H3/t3-,4-,5+,6-,7-/m1/s1
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Article
PubMed
n/an/a 2.80E+4n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase


(Homo sapiens (Human))
BDBM50122955
PNG
(2-(4,6-Difluoro-indan-1-ylidene)-acetamide | CHEMB...)
Show SMILES NC(=O)\C=C1/CCc2c1cc(F)cc2F
Show InChI InChI=1S/C11H9F2NO/c12-7-4-9-6(3-11(14)15)1-2-8(9)10(13)5-7/h3-5H,1-2H2,(H2,14,15)/b6-3+
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UniChem

Patents

Article
PubMed
n/an/a 3.00E+4n/an/an/an/an/an/a



GlaxoSmithKline Research and Development

Curated by ChEMBL


Assay Description
Inhibitory concentration of the compound against lysyl oxidase


J Med Chem 46: 399-408 (2003)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232680
PNG
(CHEMBL4084804)
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n/an/a>3.10E+4n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18361
PNG
((2R,3S,4R,5R,6R)-2-butyl-6-(hydroxymethyl)piperidi...)
Show SMILES CCCC[C@H]1N[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O
Show InChI InChI=1S/C10H21NO4/c1-2-3-4-6-8(13)10(15)9(14)7(5-12)11-6/h6-15H,2-5H2,1H3/t6-,7-,8+,9-,10-/m1/s1
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Article
PubMed
n/an/a 3.10E+4n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50232692
PNG
(CHEMBL4098672)
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n/an/a 3.50E+4n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM50408786
PNG
(CHEMBL148476)
Show SMILES NCc1ccc(N)cc1
Show InChI InChI=1S/C7H10N2/c8-5-6-1-3-7(9)4-2-6/h1-4H,5,8-9H2
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n/an/a 4.70E+4n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
alpha-Glucosidase (alpha-Glu)


(Homo sapiens (Human))
BDBM18354
PNG
((2R,3R,4R,5S)-2-(hydroxymethyl)-1-propylpiperidine...)
Show SMILES CCCN1C[C@H](O)[C@@H](O)[C@H](O)[C@H]1CO
Show InChI InChI=1S/C9H19NO4/c1-2-3-10-4-7(12)9(14)8(13)6(10)5-11/h6-9,11-14H,2-5H2,1H3/t6-,7+,8-,9-/m1/s1
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Article
PubMed
n/an/a 5.60E+4n/an/an/an/a4.537



Hokuriku University



Assay Description
Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...


Bioorg Med Chem 14: 7736-44 (2006)

More data for this
Ligand-Target Pair
Lysyl oxidase homolog 2


(Homo sapiens (Human))
BDBM10758
PNG
(14C-phenylethylamine | 2-phenylethan-1-amine | CHE...)
Show SMILES NCCc1ccccc1
Show InChI InChI=1S/C8H11N/c9-7-6-8-4-2-1-3-5-8/h1-5H,6-7,9H2
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n/an/a 6.01E+4n/an/an/an/an/an/a



PharmAkea Inc.

Curated by ChEMBL




Citation and Details
More data for this
Ligand-Target Pair
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