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Compile Data Set for Download or QSAR

Found 205 hits Enz. Inhib. hit(s) with Target = 'Menin'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 11
PNG
GoogleScholar
AffyNet 
UniChem
Article
0.440n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 34
PNG
GoogleScholar
AffyNet 
UniChem
Article
0.530n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 20
PNG
GoogleScholar
AffyNet 
UniChem
Article
0.670n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 87
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.10n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 88
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.30n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 103
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.40n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 18
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.5n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 19
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.80n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 102
PNG
GoogleScholar
AffyNet 
UniChem
Article
1.80n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 4
PNG
GoogleScholar
AffyNet 
UniChem
Article
2.20n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 76
PNG
GoogleScholar
AffyNet 
UniChem
Article
2.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 66
PNG
GoogleScholar
AffyNet 
UniChem
Article
2.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 5
PNG
GoogleScholar
AffyNet 
UniChem
Article
2.70n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 33
PNG
GoogleScholar
AffyNet 
UniChem
Article
3.20n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 9
PNG
GoogleScholar
AffyNet 
UniChem
Article
3.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 35
PNG
GoogleScholar
AffyNet 
UniChem
Article
3.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 10
PNG
GoogleScholar
AffyNet 
UniChem
Article
5n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 36
PNG
GoogleScholar
AffyNet 
UniChem
Article
5.20n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 42
PNG
GoogleScholar
AffyNet 
UniChem
Article
6.20n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 96
PNG
GoogleScholar
AffyNet 
UniChem
Article
6.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 61
PNG
GoogleScholar
AffyNet 
UniChem
Article
6.90n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 67
PNG
GoogleScholar
AffyNet 
UniChem
Article
8.10n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 62
PNG
GoogleScholar
AffyNet 
UniChem
Article
8.5n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 64
PNG
GoogleScholar
AffyNet 
UniChem
Article
8.60n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 40
PNG
GoogleScholar
AffyNet 
UniChem
Article
8.90n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 70
PNG
GoogleScholar
AffyNet 
UniChem
Article
9n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 28
PNG
GoogleScholar
AffyNet 
UniChem
Article
11n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 101
PNG
GoogleScholar
AffyNet 
UniChem
Article
11n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 21
PNG
GoogleScholar
AffyNet 
UniChem
Article
12n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 29
PNG
GoogleScholar
AffyNet 
UniChem
Article
13n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 23
PNG
GoogleScholar
AffyNet 
UniChem
Article
13n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 108
PNG
GoogleScholar
AffyNet 
UniChem
Article
15n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 53
PNG
GoogleScholar
AffyNet 
UniChem
Article
17n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 54
PNG
GoogleScholar
AffyNet 
UniChem
Article
18n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
BDBM321268
PNG
(N-[4-(benzylmethylamino)butyl]-4-chlorobenzamide |...)
GoogleScholar
AffyNet 
UniChem
Article
20n/an/an/an/an/an/an/an/a



Universita degli Studi





J Med Chem 43: 3677-87 (2000)


Article DOI: 10.1021/jm058056x
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 38
PNG
GoogleScholar
AffyNet 
UniChem
Article
21n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 39
PNG
GoogleScholar
AffyNet 
UniChem
Article
21n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 48
PNG
GoogleScholar
AffyNet 
UniChem
Article
22n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 22
PNG
GoogleScholar
AffyNet 
UniChem
Article
23n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 49
PNG
GoogleScholar
AffyNet 
UniChem
Article
25n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 1
PNG
GoogleScholar
AffyNet 
UniChem
Article
25n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 109
PNG
GoogleScholar
AffyNet 
UniChem
Article
31n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 58
PNG
GoogleScholar
AffyNet 
UniChem
Article
32n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 50
PNG
GoogleScholar
AffyNet 
UniChem
Article
37n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 41
PNG
GoogleScholar
AffyNet 
UniChem
Article
38n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 26
PNG
GoogleScholar
AffyNet 
UniChem
Article
41n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
BDBM321277
PNG
(N-[3-(benzylmethylamino)propyl]-3,5-dichlorobenzam...)
GoogleScholar
AffyNet 
UniChem
Article
48n/an/an/an/an/an/an/an/a



Universita degli Studi





J Med Chem 43: 3677-87 (2000)


Article DOI: 10.1021/jm058056x
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
BDBM321260
PNG
(N-[3-(benzylmethylamino)propyl]-4-butylbenzamide |...)
GoogleScholar
AffyNet 
UniChem
Article
49n/an/an/an/an/an/an/an/a



Universita degli Studi





J Med Chem 43: 3677-87 (2000)


Article DOI: 10.1021/jm058056x
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 24
PNG
GoogleScholar
AffyNet 
UniChem
Article
52n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
Sigma intracellular receptor 2


(Homo sapiens (Human))
US10207991, Ex. Cpd. No. 59
PNG
GoogleScholar
AffyNet 
UniChem
Article
57n/an/an/an/an/an/an/an/a



Pfizer





J Med Chem 50: 182-5 (2007)


Article DOI: 10.1021/jm060653b
More data for this
Ligand-Target Pair
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