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Compile Data Set for Download or QSAR

Found 82 hits Enz. Inhib. hit(s) with Target = 'cAMP-specific 3',5'-cyclic phosphodiesterase 4A'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285634
PNG
(3-(4-chloro-3,5-difluoro-phenyl)-N-cyclopropyl-imi...)
Show SMILES Fc1cc(cc(F)c1Cl)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a<0.488n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285598
PNG
(3-(3-chloro-4-methylphenyl)-N-[(1R,2S)-2-fluorocyc...)
Show SMILES Cc1ccc(cc1Cl)-c1c(nc2cccnn12)C(=O)N[C@@H]1C[C@@H]1F
GoogleScholar
AffyNet 
UniChem
Article
n/an/a<0.669n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285537
PNG
(3-(4-chloro-3-fluoro-phenyl)-N-cyclopropyl-imidazo...)
Show SMILES Fc1cc(ccc1Cl)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 1.51n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285534
PNG
(3-(4-Chloro-3-fluorophenyl)-N-(1-methyl-1H-pyrazol...)
Show SMILES Cn1cc(NC(=O)c2nc3cccnn3c2-c2ccc(Cl)c(F)c2)cn1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 2.77n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285572
PNG
(3-(4-chloro-3-fluorophenyl)-N-[(1R,2S)-2-fluorocyc...)
Show SMILES F[C@H]1C[C@H]1NC(=O)c1nc2cccnn2c1-c1ccc(Cl)c(F)c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 2.91n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285568
PNG
(N-cyclopropyl-3-(3-fluoro-4-methylphenyl)imidazo[1...)
Show SMILES Cc1ccc(cc1F)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 3.13n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285556
PNG
(3-(4-chloro-3-fluorophenyl)-N-propylimidazo[1,2-b]...)
Show SMILES CCCNC(=O)c1nc2cccnn2c1-c1ccc(Cl)c(F)c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 3.48n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285536
PNG
(3-(4-Chloro-2,5-difluorophenyl)-N-cyclopropylimida...)
Show SMILES Fc1cc(-c2c(nc3cccnn23)C(=O)NC2CC2)c(F)cc1Cl
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 3.83n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285576
PNG
(US10077269, Example 49 | US9598421, Example 49 | a...)
Show SMILES Cc1ccc(cc1Cl)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 4.16n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285626
PNG
(3-(4-chloro-2,5-difluoro-phenyl)-N-ethylimidazo[1,...)
Show SMILES CCNC(=O)c1nc2cccnn2c1-c1cc(F)c(Cl)cc1F
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 4.58n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285551
PNG
(4-[2-(azetidin-1-ylcarbonyl)imidazo[1,2-b]pyridazi...)
Show SMILES Fc1cc(-c2c(nc3cccnn23)C(=O)N2CCC2)c(F)cc1C#N
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 5.04n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285540
PNG
(US10077269, Example 13 | US9598421, Example 13 | a...)
Show SMILES Fc1cc(ccc1Cl)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 5.13n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285627
PNG
(3-(4-chloro-5-fluoro-2-methylphenyl)-N-(propan-2-y...)
Show SMILES CC(C)NC(=O)c1nc2cccnn2c1-c1cc(F)c(Cl)cc1C
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 5.48n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285622
PNG
(3-(4-cyano-2,5-difluorophenyl)-N-cyclopropylimidaz...)
Show SMILES Fc1cc(-c2c(nc3cccnn23)C(=O)NC2CC2)c(F)cc1C#N
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 5.52n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285616
PNG
(US10077269, Example 86 | US9598421, Example 86 | a...)
Show SMILES FC1(F)Oc2ccc(cc2O1)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 5.83n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285613
PNG
(US10077269, Example 83 | US9598421, Example 83 | a...)
Show SMILES Clc1ccc(cc1Cl)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 6.21n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285547
PNG
(4-[2-(azetidin-1-ylcarbonyl)imidazo[1,2-b]pyridazi...)
Show SMILES Cc1cc(C#N)c(F)cc1-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 6.70n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285603
PNG
(US10077269, Example 76 | US9598421, Example 76 | a...)
Show SMILES FC(F)Oc1cc(ccn1)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 7.09n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285574
PNG
(US10077269, Example 47 | US9598421, Example 47 | a...)
Show SMILES Fc1cc(cc(F)c1Cl)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 7.37n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285611
PNG
(3-(4-chloro-3-fluorophenyl)-N-ethylimidazo[1,2-b]p...)
Show SMILES CCNC(=O)c1nc2cccnn2c1-c1ccc(Cl)c(F)c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 7.86n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285602
PNG
(N-cyclopropyl-3-[2-(difluoro-methoxy)pyridin-4-yl]...)
Show SMILES FC(F)Oc1cc(ccn1)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 10.5n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285595
PNG
(3-(4-chloro-2-fluorophenyl)-N-[(1R,2S)-2-fluorocyc...)
Show SMILES F[C@H]1C[C@H]1NC(=O)c1nc2cccnn2c1-c1ccc(Cl)cc1F
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 10.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285529
PNG
(3-(4-Chlorophenyl)-N-cyclopropylimidazo[1,2-b]pyri...)
Show SMILES Clc1ccc(cc1)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 10.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285557
PNG
(3-(4-chlorophenyl)-N-(2-methylcyclopropyl)imidazo[...)
Show SMILES CC1CC1NC(=O)c1nc2cccnn2c1-c1ccc(Cl)cc1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 11.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285612
PNG
(3-(4-chloro-3-fluorophenyl)-N-(1H-pyrazol-4-yl)imi...)
Show SMILES Fc1cc(ccc1Cl)-c1c(nc2cccnn12)C(=O)Nc1cn[nH]c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 12n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285621
PNG
(US10077269, Example 91 | US9598421, Example 91 | a...)
Show SMILES Fc1cc(-c2c(nc3cccnn23)C(=O)N2CCC2)c(F)cc1Cl
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 12.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285530
PNG
(Azetidin-1-yl[3-(3,5-difluoro-4-methoxyphenyl)imid...)
Show SMILES COc1c(F)cc(cc1F)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 12.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285539
PNG
(3-(4-chloro-2-methyl-phenyl)-N-cyclopropyl-imidazo...)
Show SMILES Cc1cc(Cl)ccc1-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 14.4n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285566
PNG
(3-(1,3-benzoxazol-5-yl)-N-cyclopropylimidazo[1,2-b...)
Show SMILES O=C(NC1CC1)c1nc2cccnn2c1-c1ccc2ocnc2c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 14.8n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285550
PNG
(4-[2-(azetidin-1-ylcarbonyl)imidazo[1,2-b]pyridazi...)
Show SMILES Fc1cc(ccc1C#N)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 15.1n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285573
PNG
(3-(4-chlorophenyl)-N-[(1R,2S)-2-fluorocyclopro-pyl...)
Show SMILES F[C@H]1C[C@H]1NC(=O)c1nc2cccnn2c1-c1ccc(Cl)cc1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 15.2n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285555
PNG
(3-(3,5-dichlorophenyl)-N-propylimidazo[1,2-b]pyrid...)
Show SMILES CCCNC(=O)c1nc2cccnn2c1-c1cc(Cl)cc(Cl)c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 15.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285614
PNG
(US10077269, Example 84 | US9598421, Example 84 | a...)
Show SMILES Clc1cccc(c1)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 16.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285546
PNG
(3-(4-cyano-5-fluoro-2-methylphenyl)-N-cyclo-propyl...)
Show SMILES Cc1cc(C#N)c(F)cc1-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 16.9n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285580
PNG
(US10077269, Example 53 | US9598421, Example 53 | a...)
Show SMILES Cc1cc(cc(C)c1F)-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 17.8n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285567
PNG
(3-(4-chloro-2-fluorophenyl)-N-cyclopropylimidazo[1...)
Show SMILES Fc1cc(Cl)ccc1-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 19.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285629
PNG
(3-(4-cyano-5-fluoro-2-methylphenyl)-N-(propan-2-yl...)
Show SMILES CC(C)NC(=O)c1nc2cccnn2c1-c1cc(F)c(cc1C)C#N
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 19.8n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285535
PNG
(Azetidin-1-yl[3-(pyrazolo[1,5-a]pyridin-6-yl)imida...)
Show SMILES O=C(N1CCC1)c1nc2cccnn2c1-c1ccc2ccnn2c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 20n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285620
PNG
(3-(4-cyano-3-fluorophenyl)-N-cyclopropylimidazo[1,...)
Show SMILES Fc1cc(ccc1C#N)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 21.4n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285583
PNG
(US10077269, Example 56 | US9598421, Example 56 | a...)
Show SMILES Cc1cc(Cl)ccc1-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 22.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285563
PNG
(3-(3-chlorophenyl)-N-cyclopropylimidazo[1,2-b]pyri...)
Show SMILES Clc1cccc(c1)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 23.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285579
PNG
(US10077269, Example 52 | US9598421, Example 52 | a...)
Show SMILES Fc1cc(Cl)ccc1-c1c(nc2cccnn12)C(=O)N1CCC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 24.3n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285624
PNG
(3-(4-chloro-3-fluorophenyl)-N-methylimidazo[1,2-b]...)
Show SMILES CNC(=O)c1nc2cccnn2c1-c1ccc(Cl)c(F)c1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 24.9n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285615
PNG
(3-(4-chlorophenyl)-N-ethylimidazo[1,2-b]pyridazine...)
Show SMILES CCNC(=O)c1nc2cccnn2c1-c1ccc(Cl)cc1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 25.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285628
PNG
(3-(4-cyano-5-fluoro-2-methyl-phenyl)-N-ethylimidaz...)
Show SMILES CCNC(=O)c1nc2cccnn2c1-c1cc(F)c(cc1C)C#N
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UniChem
Article
n/an/a 26.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285549
PNG
(N-cyclopropyl-3-(pyrazolo[1,5-a]pyridin-6-yl)imida...)
Show SMILES O=C(NC1CC1)c1nc2cccnn2c1-c1ccc2ccnn2c1
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UniChem
Article
n/an/a 27.6n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285577
PNG
(US10077269, Example 50 | US9598421, Example 50 | a...)
Show SMILES O=C(N1CCC1)c1nc2cccnn2c1-c1ccc2OCCc2c1
GoogleScholar
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UniChem
Article
n/an/a 28.1n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285561
PNG
(3-(3-chloro-5-fluorophenyl)-N-propylimidazo[1,2-b]...)
Show SMILES CCCNC(=O)c1nc2cccnn2c1-c1cc(F)cc(Cl)c1
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UniChem
Article
n/an/a 29.5n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285562
PNG
(3-(3-chloro-5-fluorophenyl)-N-cyclopropylimidazo[1...)
Show SMILES Fc1cc(Cl)cc(c1)-c1c(nc2cccnn12)C(=O)NC1CC1
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 35.7n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4A isoform 3


(Homo sapiens (Human))
BDBM285597
PNG
(3-(4-chloro-2-methylphenyl)-N-[(1R,2S)-2-fluorocyc...)
Show SMILES Cc1cc(Cl)ccc1-c1c(nc2cccnn12)C(=O)N[C@@H]1C[C@@H]1F
GoogleScholar
AffyNet 
UniChem
Article
n/an/a 36.4n/an/an/an/an/an/a



SUGEN, Inc.





J Med Chem 46: 1116-9 (2003)

More data for this
Ligand-Target Pair
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