Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM98008 (US8481743, 4) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 19.2 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM98007 (US8481743, 3) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 36.1 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM98009 (US8481743, 1) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 82.8 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM98006 (US8481743, 2) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 331 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM98006 (US8481743, 2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM98009 (US8481743, 1) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM98008 (US8481743, 4) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Homo sapiens (Human)) | BDBM98007 (US8481743, 3) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Purdue Pharma L.P. US Patent | Assay Description Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor. | US Patent US8481743 (2013) BindingDB Entry DOI: 10.7270/Q2BK19Z7 | |||||||||||
More data for this Ligand-Target Pair |