Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prolyl endopeptidase FAP (Homo sapiens (Human)) | BDBM103917 (US8562945, 253) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit separase enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl endopeptidase FAP (Homo sapiens (Human)) | BDBM103918 (US8562945, 254) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit separase enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103909 (JNK3 inhibitor 6 | US8562945, 242) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103908 (JNK3 inhibitor 5 | US8562945, 241) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103911 (JNK3 inhibitor 8 | US8562945, 246) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 42 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103915 (US8562945, 250) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 130 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103911 (JNK3 inhibitor 8 | US8562945, 246) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 140 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103909 (JNK3 inhibitor 6 | US8562945, 242) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 170 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103914 (US8562945, 249) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 189 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103913 (US8562945, 248) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 260 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103912 (US8562945, 247) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 305 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103914 (US8562945, 249) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 405 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103908 (JNK3 inhibitor 5 | US8562945, 241) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 445 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 9 (Homo sapiens (Human)) | BDBM103910 (JNK3 inhibitor 7 | US8562945, 243) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 564 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103910 (JNK3 inhibitor 7 | US8562945, 243) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 652 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103915 (US8562945, 250) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 669 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103913 (US8562945, 248) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 770 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carbonic anhydrase 2 (Homo sapiens (Human)) | BDBM103912 (US8562945, 247) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.16E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit carbonic anhydrase isozymes II and IX in vito. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl endopeptidase FAP (Homo sapiens (Human)) | BDBM103916 (US8562945, 252) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.53E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit separase enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM103917 (US8562945, 253) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit DPPIV enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM103916 (US8562945, 252) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.96E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit DPPIV enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM103918 (US8562945, 254) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.54E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Molecular Insight Pharmaceuticals, Inc. US Patent | Assay Description Compounds were tested for their ability to inhibit DPPIV enzyme. | US Patent US8562945 (2013) BindingDB Entry DOI: 10.7270/Q2XP73KD | |||||||||||
More data for this Ligand-Target Pair |