Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Regulator of G-protein signaling 4 (Homo sapiens (Human)) | BDBM50384774 (CHEMBL1917204 | US20230414581, Compound 6) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 19 (Homo sapiens (Human)) | BDBM50384774 (CHEMBL1917204 | US20230414581, Compound 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 16 (Homo sapiens (Human)) | BDBM50384774 (CHEMBL1917204 | US20230414581, Compound 6) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM50384774 (CHEMBL1917204 | US20230414581, Compound 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 4 (Homo sapiens (Human)) | BDBM136369 (US8865750, CCG- 203780) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 3.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 4 (Homo sapiens (Human)) | BDBM50384773 (CHEMBL2037371) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 9.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM136368 (US8865750, CCG- 203778) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM50384773 (CHEMBL2037371) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 4 (Homo sapiens (Human)) | BDBM136368 (US8865750, CCG- 203778) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM136369 (US8865750, CCG- 203780) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Regents of The University of Michigan; The University of Bath US Patent | Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp... | US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC | |||||||||||
More data for this Ligand-Target Pair |