Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM152814 (US8993575, 4) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.510 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM152813 (US8993575, 3) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.27 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50130293 (7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB US Patent | n/a | n/a | 3.35 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM152813 (US8993575, 3) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8.82 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM50130293 (7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 11.5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM152814 (US8993575, 4) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 12.7 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM152816 (US8993575, 6) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 15.1 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM152816 (US8993575, 6) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 19.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM152815 (US8993575, 5) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 26.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM152815 (US8993575, 5) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 62.5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (Rattus norvegicus (rat)) | BDBM152817 (US8993575, 12) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 122 | n/a | n/a | n/a | n/a | 7.5 | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Materials for the Receptor Binding AssayIsotope ligand [3H]-Ketanserin (67.0 Ci/mmol) was purchased from PerkinElmer Company; Methysergide was purcha... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM152817 (US8993575, 12) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
Huazhong University of Science & Technology; NHWA Pharma Corporation US Patent | Assay Description Isotope ligand 3H-8-OH-DPAT (67.0 Ci/mmol) was purchased from PerkinElmer Company; 5-HT was purchased from RBI Company; GF/C glass fiber filter paper... | US Patent US8993575 (2015) BindingDB Entry DOI: 10.7270/Q2RX99TN | |||||||||||
More data for this Ligand-Target Pair |