Affinity Data by Patent

Patent code US9114126

Found 10 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM50292546 (3,4,5,6-tetrahydroxyxanthone \| CHEMBL477921 \| US91...) Show SMILES Oc1ccc2c(oc3c(O)c(O)ccc3c2=O)c1O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174833 (3,4,5-Trihydroxy xanthone (1) \| US9114126, MB5) Show SMILES Oc1ccc2c(oc3c(O)cccc3c2=O)c1O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM50292547 (1,3,5,6-tetrahydroxyxanthone \| 1,3,5,6-tetrahydrox...) Show SMILES Oc1cc(O)c2c(c1)oc1c(O)c(O)ccc1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	6.00E+4	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM50155436 (1,3,5-Trihydroxy-xanthen-9-one \| CHEMBL365234 \| US...) Show SMILES Oc1cc(O)c2c(c1)oc1c(O)cccc1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	6.50E+4	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM50269645 (3,4-dihydroxyxanthone \| CHEMBL446323 \| US9114126, ...) Show SMILES Oc1ccc2c(oc3ccccc3c2=O)c1O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174835 (US9114126, 2027BA1) Show SMILES COc1cc(O)c2c(c1)oc1ccc(O)c(OC)c1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	KEGG PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174834 (US9114126, MB8) Show SMILES COc1ccc2c(c1)oc1c(OC)c(OC)ccc1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174836 (US9114126, 2027BA2) Show SMILES COc1cc(O)c2c(c1)oc1ccc(OC)c(O)c1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase MCE KEGG PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174837 (US9114126, C-017) Show SMILES COc1ccc2oc3cc(OC)c(OC)c(OC)c3c(=O)c2c1 Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair
Potassium-transporting ATPase alpha chain 1 (Sus scrofa (Pig))	BDBM174832 (US9114126, MB1) Show SMILES Oc1cc(O)c2c(c1)oc1ccccc1c2=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.4	37
THE UNIVERSITY OF TOLEDO US Patent					Assay Description The purified Na/K-ATPase was prepared from pig kidney. The specific activities of Na/K-ATPase of various kidney preparations were in the range of 900...				US Patent US9114126 (2015) BindingDB Entry DOI: 10.7270/Q2Z31XFQ
THE UNIVERSITY OF TOLEDO US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%