Affinity Data by Patent

Patent code US9120786

Found 14 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177783 (US10000475, Compound 12 \| US9120786, 12) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	243	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177773 (US10000475, Compound 2 \| US9120786, 2) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	326	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177781 (US10000475, Compound 10 \| US9120786, 10) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	353	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177780 (US10000475, Compound 9 \| US9120786, 9) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	596	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177776 (US10000475, Compound 5 \| US9120786, 5) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	645	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177777 (US10000475, Compound 6 \| US9120786, 6) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.80E+3	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177772 (US10000475, Compound 1 \| US9120786, 1) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.25E+3	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177779 (US10000475, Compound 8 \| US9120786, 8) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	8.09E+3	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177785 (US10000475, Compound 14 \| US9120786, 14) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177774 (US10000475, Compound 3 \| US9120786, 3) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177784 (US10000475, Compound 13 \| US9120786, 13) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177775 (US10000475, Compound 4 \| US9120786, 4) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177782 (US10000475, Compound 11 \| US9120786, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair
Sodium channel protein type 9 subunit alpha (Homo sapiens (Human))	BDBM177778 (US10000475, Compound 7 \| US9120786, 7) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	37
Purdue Pharma, L.P. US Patent					Assay Description FLIPRTETRA Sodium Dye Assay with KCl: Cells were prepared by plating the recombinant HEK293 cells or other host cells expressing either recombinant o...				US Patent US9120786 (2015) BindingDB Entry DOI: 10.7270/Q25D8QKN
Purdue Pharma, L.P. US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%