Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM50310923 (CHEMBL1077943 | US9120807, 6 | {6-Methylamino-2-[(...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM50310925 (CHEMBL1081160 | US9120807, 7 | {6-dimethylamino-2-...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM50310924 (CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM50310922 (CHEMBL1080241 | US9120807, 9 | {6-Amino-2-[(pyridi...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50310925 (CHEMBL1081160 | US9120807, 7 | {6-dimethylamino-2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 19.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM50310923 (CHEMBL1077943 | US9120807, 6 | {6-Methylamino-2-[(...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 22.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM177999 (US9120807, 11) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 36.7 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM50310924 (CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 37.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM177998 (US9120807, 10) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 52.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50310923 (CHEMBL1077943 | US9120807, 6 | {6-Methylamino-2-[(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 57.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2b (Homo sapiens (Human)) | BDBM178000 (US9120807, 12) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 68.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50310924 (CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 118 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM50310925 (CHEMBL1081160 | US9120807, 7 | {6-dimethylamino-2-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM177998 (US9120807, 10) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 161 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM177999 (US9120807, 11) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 216 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM50310922 (CHEMBL1080241 | US9120807, 9 | {6-Amino-2-[(pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 233 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM178000 (US9120807, 12) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 256 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50310923 (CHEMBL1077943 | US9120807, 6 | {6-Methylamino-2-[(...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 277 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM178000 (US9120807, 12) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 308 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50310925 (CHEMBL1081160 | US9120807, 7 | {6-dimethylamino-2-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 318 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM177999 (US9120807, 11) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 361 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50310924 (CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 726 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM177998 (US9120807, 10) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 747 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM178000 (US9120807, 12) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 828 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50310922 (CHEMBL1080241 | US9120807, 9 | {6-Amino-2-[(pyridi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50310922 (CHEMBL1080241 | US9120807, 9 | {6-Amino-2-[(pyridi...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM177999 (US9120807, 11) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM177998 (US9120807, 10) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vernalis (R&D) Ltd. US Patent | Assay Description The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique... | US Patent US9120807 (2015) BindingDB Entry DOI: 10.7270/Q2NG4PDH | |||||||||||
More data for this Ligand-Target Pair |