Affinity Data by Patent

Patent code US9150583

Found 8 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184568 (US9150583, 5) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	9	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184566 (US9150583, 3) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184570 (US9150583, 7) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184564 (US9150583, 1) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184565 (US9150583, 2) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184569 (US9150583, 6) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184567 (US9150583, 4) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	90	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM184571 (US9150583, 8) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	37
Boehringer Ingelheim International GmbH US Patent					Assay Description CETP inhibitory activity of compounds of the present invention can be determined in a fluorometric assay purchased from Roar Biomedical, Inc. (New Yo...				US Patent US9150583 (2015) BindingDB Entry DOI: 10.7270/Q2Z89B5V
Boehringer Ingelheim International GmbH US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%