Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443628 (CHEMBL3092468 | US9174993, 35 | US9221828, 35) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443633 (CHEMBL3092463 | US9174993, 7 | US9221828, 7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443634 (CHEMBL3092462 | US9174993, 6 | US9221828, 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443630 (CHEMBL3092466 | US9174993, 15 | US9221828, 15) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043873 (CHEMBL3356059 | US9174993, 11 | US9221828, 11) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043783 (CHEMBL3356053 | US9174993, 46 | US9221828, 46) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443629 (CHEMBL3092467 | US9174993, 16 | US9221828, 16) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443636 (CHEMBL3092460 | US9174993, 1 | US9221828, 1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043874 (CHEMBL3356060 | US9174993, 13 | US9221828, 13) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443631 (CHEMBL3092465 | US9174993, 14 | US9221828, 14) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043784 (CHEMBL3356054 | US9174993, 9 | US9221828, 9) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443632 (CHEMBL3092464 | US9174993, 12 | US9221828, 12) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50443635 (CHEMBL3092461 | US9174993, 5 | US9221828, 5) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043872 (CHEMBL3356058 | US9174993, 10 | US9221828, 10) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043916 (CHEMBL3356041 | US9174993, 64) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043921 (CHEMBL3356047 | US9174993, 58) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM189809 (US9174993, 61) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043917 (CHEMBL3356042 | US9174993, 63) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043920 (CHEMBL3356046 | US9174993, 59) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM189808 (US9174993, 60) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM189807 (US9174993, 45 | US9221828, 45) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043899 (CHEMBL3356040 | US9174993, 8 | US9221828, 8) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 196 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM189805 (US9174993, 42 | US9221828, 42) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 413 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043871 (CHEMBL3356057 | US9174993, 4 | US9221828, 4) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 419 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043786 (CHEMBL3356055 | US9174993, 2 | US9221828, 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 439 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM50043787 (CHEMBL3356056 | US9174993, 3 | US9221828, 3) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 496 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase Sgk1 (Homo sapiens (Human)) | BDBM189806 (US9174993, 43) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
SANOFI US Patent | Assay Description The compounds were tested for serum and glucocorticoid-regulated kinase 1 (SGK-1) inhibitory activity in a substrate phosphorylation assay designed t... | US Patent US9174993 (2015) BindingDB Entry DOI: 10.7270/Q2MK6BPF | |||||||||||
More data for this Ligand-Target Pair |