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Patent code US9216962

Compile Data Set for Download or QSAR

Found 216 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197350
PNG
(US9216962, CFH395-C)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C17H22N4O3S2/c22-12(21-24)5-3-1-2-4-8-18-15(23)13-14(11-6-7-11)26-17(20-13)16-19-9-10-25-16/h9-11,24H,1-8H2,(H,18,23)(H,21,22)
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n/an/a 10n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197350
PNG
(US9216962, CFH395-C)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C17H22N4O3S2/c22-12(21-24)5-3-1-2-4-8-18-15(23)13-14(11-6-7-11)26-17(20-13)16-19-9-10-25-16/h9-11,24H,1-8H2,(H,18,23)(H,21,22)
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n/an/a 10n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197362
PNG
(US9216962, CFH449-H)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
Show InChI InChI=1S/C21H28N4O3S2/c26-16(25-28)9-3-1-2-6-12-22-19(27)17-18(13-10-11-13)30-21(24-17)20-23-14-7-4-5-8-15(14)29-20/h13,28H,1-12H2,(H,22,27)(H,25,26)
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n/an/a 11n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197363
PNG
(US9216962, CFH443-5)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccccc1
Show InChI InChI=1S/C21H22N4O3S2/c26-16(25-28)8-4-5-11-22-19(27)17-18(14-9-10-14)30-21(24-17)20-23-12-15(29-20)13-6-2-1-3-7-13/h1-3,6-7,12,14,28H,4-5,8-11H2,(H,22,27)(H,25,26)
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n/an/a 11n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020910
PNG
(CHEMBL3287268 | US9216962, CFH395)
Show SMILES CC(C)\C=C\c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C17H22N4O3S2/c1-11(2)6-7-12-14(20-17(26-12)16-19-9-10-25-16)15(23)18-8-4-3-5-13(22)21-24/h6-7,9-11,24H,3-5,8H2,1-2H3,(H,18,23)(H,21,22)/b7-6+
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n/an/a 13n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197362
PNG
(US9216962, CFH449-H)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
Show InChI InChI=1S/C21H28N4O3S2/c26-16(25-28)9-3-1-2-6-12-22-19(27)17-18(13-10-11-13)30-21(24-17)20-23-14-7-4-5-8-15(14)29-20/h13,28H,1-12H2,(H,22,27)(H,25,26)
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n/an/a 16n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197350
PNG
(US9216962, CFH395-C)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C17H22N4O3S2/c22-12(21-24)5-3-1-2-4-8-18-15(23)13-14(11-6-7-11)26-17(20-13)16-19-9-10-25-16/h9-11,24H,1-8H2,(H,18,23)(H,21,22)
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n/an/a 20n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197366
PNG
(US9216962, CFH401)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nccs2)cc1
Show InChI InChI=1S/C18H16N4O3S2/c23-15(22-25)12-3-1-10(2-4-12)9-20-16(24)13-14(11-5-6-11)27-18(21-13)17-19-7-8-26-17/h1-4,7-8,11,25H,5-6,9H2,(H,20,24)(H,22,23)
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n/an/a 20n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197343
PNG
(US9216962, CFH424)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C19H28N4O3S2/c1-13(2)12-14-16(22-19(28-14)18-21-10-11-27-18)17(25)20-9-7-5-3-4-6-8-15(24)23-26/h10-11,13,26H,3-9,12H2,1-2H3,(H,20,25)(H,23,24)
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n/an/a 21n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020908
PNG
(CHEMBL3287266 | US9216962, CFH367)
Show SMILES C\C=C\c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C15H18N4O3S2/c1-2-5-10-12(18-15(24-10)14-17-8-9-23-14)13(21)16-7-4-3-6-11(20)19-22/h2,5,8-9,22H,3-4,6-7H2,1H3,(H,16,21)(H,19,20)/b5-2+
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n/an/a 22n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197356
PNG
(US9216962, CFH421-C)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
Show InChI InChI=1S/C19H24N4O3S2/c24-14(23-26)7-3-4-10-20-17(25)15-16(11-8-9-11)28-19(22-15)18-21-12-5-1-2-6-13(12)27-18/h11,26H,1-10H2,(H,20,25)(H,23,24)
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n/an/a 25n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197366
PNG
(US9216962, CFH401)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nccs2)cc1
Show InChI InChI=1S/C18H16N4O3S2/c23-15(22-25)12-3-1-10(2-4-12)9-20-16(24)13-14(11-5-6-11)27-18(21-13)17-19-7-8-26-17/h1-4,7-8,11,25H,5-6,9H2,(H,20,24)(H,22,23)
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n/an/a 30n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020896
PNG
(CHEMBL3287254 | US9216962, CFH383)
Show SMILES CCCCc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C16H22N4O3S2/c1-2-3-6-11-13(19-16(25-11)15-18-9-10-24-15)14(22)17-8-5-4-7-12(21)20-23/h9-10,23H,2-8H2,1H3,(H,17,22)(H,20,21)
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n/an/a 31n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020894
PNG
(CHEMBL3287252 | US9216962, CFH355)
Show SMILES CCc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C14H18N4O3S2/c1-2-9-11(17-14(23-9)13-16-7-8-22-13)12(20)15-6-4-3-5-10(19)18-21/h7-8,21H,2-6H2,1H3,(H,15,20)(H,18,19)
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n/an/a 31n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197363
PNG
(US9216962, CFH443-5)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccccc1
Show InChI InChI=1S/C21H22N4O3S2/c26-16(25-28)8-4-5-11-22-19(27)17-18(14-9-10-14)30-21(24-17)20-23-12-15(29-20)13-6-2-1-3-7-13/h1-3,6-7,12,14,28H,4-5,8-11H2,(H,22,27)(H,25,26)
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n/an/a 32n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197341
PNG
(US9216962, CFH396)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C17H24N4O3S2/c1-11(2)10-12-14(20-17(26-12)16-19-8-9-25-16)15(23)18-7-5-3-4-6-13(22)21-24/h8-9,11,24H,3-7,10H2,1-2H3,(H,18,23)(H,21,22)
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n/an/a 35n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197349
PNG
(US9216962, CFH381-C)
Show SMILES ONC(=O)CCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C16H20N4O3S2/c21-11(20-23)4-2-1-3-7-17-14(22)12-13(10-5-6-10)25-16(19-12)15-18-8-9-24-15/h8-10,23H,1-7H2,(H,17,22)(H,20,21)
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n/an/a 37n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197366
PNG
(US9216962, CFH401)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nccs2)cc1
Show InChI InChI=1S/C18H16N4O3S2/c23-15(22-25)12-3-1-10(2-4-12)9-20-16(24)13-14(11-5-6-11)27-18(21-13)17-19-7-8-26-17/h1-4,7-8,11,25H,5-6,9H2,(H,20,24)(H,22,23)
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n/an/a 42n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197345
PNG
(US9216962, CFH430)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1\C=C\c1ccccc1)-c1nccs1
Show InChI InChI=1S/C20H20N4O3S2/c25-16(24-27)8-4-5-11-21-18(26)17-15(10-9-14-6-2-1-3-7-14)29-20(23-17)19-22-12-13-28-19/h1-3,6-7,9-10,12-13,27H,4-5,8,11H2,(H,21,26)(H,24,25)/b10-9+
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n/an/a 47n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020890
PNG
(CHEMBL3287250 | US9216962, CFH382)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C16H22N4O3S2/c1-10(2)9-11-13(19-16(25-11)15-18-7-8-24-15)14(22)17-6-4-3-5-12(21)20-23/h7-8,10,23H,3-6,9H2,1-2H3,(H,17,22)(H,20,21)
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n/an/a 47n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197362
PNG
(US9216962, CFH449-H)
Show SMILES ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
Show InChI InChI=1S/C21H28N4O3S2/c26-16(25-28)9-3-1-2-6-12-22-19(27)17-18(13-10-11-13)30-21(24-17)20-23-14-7-4-5-8-15(14)29-20/h13,28H,1-12H2,(H,22,27)(H,25,26)
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n/an/a 49n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197355
PNG
(US9216962, CFH395-M)
Show SMILES Cc1nc(sc1C)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C17H22N4O3S2/c1-9-10(2)25-16(19-9)17-20-13(14(26-17)11-6-7-11)15(23)18-8-4-3-5-12(22)21-24/h11,24H,3-8H2,1-2H3,(H,18,23)(H,21,22)
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n/an/a 50n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020905
PNG
(CHEMBL3287263 | US9216962, CFH461)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1CCOCc1ccccc1)-c1nccs1
Show InChI InChI=1S/C21H24N4O4S2/c26-17(25-28)8-4-5-10-22-19(27)18-16(31-21(24-18)20-23-11-13-30-20)9-12-29-14-15-6-2-1-3-7-15/h1-3,6-7,11,13,28H,4-5,8-10,12,14H2,(H,22,27)(H,25,26)
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n/an/a 50n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197353
PNG
(US9216962, CFH381-B)
Show SMILES Cc1csc(n1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C16H20N4O3S2/c1-9-8-24-15(18-9)16-19-12(13(25-16)10-5-6-10)14(22)17-7-3-2-4-11(21)20-23/h8,10,23H,2-7H2,1H3,(H,17,22)(H,20,21)
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n/an/a 50n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197361
PNG
(US9216962, CFH407-C)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc(cs1)C1CC1
Show InChI InChI=1S/C18H22N4O3S2/c23-13(22-25)3-1-2-8-19-16(24)14-15(11-6-7-11)27-18(21-14)17-20-12(9-26-17)10-4-5-10/h9-11,25H,1-8H2,(H,19,24)(H,22,23)
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n/an/a 52n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197349
PNG
(US9216962, CFH381-C)
Show SMILES ONC(=O)CCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C16H20N4O3S2/c21-11(20-23)4-2-1-3-7-17-14(22)12-13(10-5-6-10)25-16(19-12)15-18-8-9-24-15/h8-10,23H,1-7H2,(H,17,22)(H,20,21)
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n/an/a 52n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197364
PNG
(US9216962, CFH443-4)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc(cs1)-c1ccccc1
Show InChI InChI=1S/C21H22N4O3S2/c26-16(25-28)8-4-5-11-22-19(27)17-18(14-9-10-14)30-21(24-17)20-23-15(12-29-20)13-6-2-1-3-7-13/h1-3,6-7,12,14,28H,4-5,8-11H2,(H,22,27)(H,25,26)
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n/an/a 56n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM50020915
PNG
(CHEMBL3287008 | US9216962, CFH412-S)
Show SMILES CC(C)[C@H](NC(=O)c1csc(n1)-c1cscn1)C(=O)OC\C=C\CCS |r|
Show InChI InChI=1S/C17H21N3O3S3/c1-11(2)14(17(22)23-6-4-3-5-7-24)20-15(21)12-9-26-16(19-12)13-8-25-10-18-13/h3-4,8-11,14,24H,5-7H2,1-2H3,(H,20,21)/b4-3+/t14-/m0/s1
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n/an/a 58n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020904
PNG
(CHEMBL3287262 | US9216962, CFH417)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1Cc1ccccc1)-c1nccs1
Show InChI InChI=1S/C19H20N4O3S2/c24-15(23-26)8-4-5-9-20-17(25)16-14(12-13-6-2-1-3-7-13)28-19(22-16)18-21-10-11-27-18/h1-3,6-7,10-11,26H,4-5,8-9,12H2,(H,20,25)(H,23,24)
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n/an/a 58n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197353
PNG
(US9216962, CFH381-B)
Show SMILES Cc1csc(n1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C16H20N4O3S2/c1-9-8-24-15(18-9)16-19-12(13(25-16)10-5-6-10)14(22)17-7-3-2-4-11(21)20-23/h8,10,23H,2-7H2,1H3,(H,17,22)(H,20,21)
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n/an/a 60n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197356
PNG
(US9216962, CFH421-C)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
Show InChI InChI=1S/C19H24N4O3S2/c24-14(23-26)7-3-4-10-20-17(25)15-16(11-8-9-11)28-19(22-15)18-21-12-5-1-2-6-13(12)27-18/h11,26H,1-10H2,(H,20,25)(H,23,24)
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n/an/a 63n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197354
PNG
(US9216962, CFH381-M)
Show SMILES Cc1cnc(s1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C16H20N4O3S2/c1-9-8-18-15(24-9)16-19-12(13(25-16)10-5-6-10)14(22)17-7-3-2-4-11(21)20-23/h8,10,23H,2-7H2,1H3,(H,17,22)(H,20,21)
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n/an/a 64n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197351
PNG
(US9216962, CFH409-C)
Show SMILES ONC(=O)CCCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C18H24N4O3S2/c23-13(22-25)6-4-2-1-3-5-9-19-16(24)14-15(12-7-8-12)27-18(21-14)17-20-10-11-26-17/h10-12,25H,1-9H2,(H,19,24)(H,22,23)
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n/an/a 64n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020897
PNG
(CHEMBL3287255 | US9216962, CFH367-C)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C15H18N4O3S2/c20-10(19-22)3-1-2-6-16-13(21)11-12(9-4-5-9)24-15(18-11)14-17-7-8-23-14/h7-9,22H,1-6H2,(H,16,21)(H,19,20)
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n/an/a 65n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197343
PNG
(US9216962, CFH424)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C19H28N4O3S2/c1-13(2)12-14-16(22-19(28-14)18-21-10-11-27-18)17(25)20-9-7-5-3-4-6-8-15(24)23-26/h10-11,13,26H,3-9,12H2,1-2H3,(H,20,25)(H,23,24)
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n/an/a 73n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197365
PNG
(US9216962, CFH455-C)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nc3CCCCc3s2)cc1
Show InChI InChI=1S/C22H22N4O3S2/c27-19(26-29)14-7-5-12(6-8-14)11-23-20(28)17-18(13-9-10-13)31-22(25-17)21-24-15-3-1-2-4-16(15)30-21/h5-8,13,29H,1-4,9-11H2,(H,23,28)(H,26,27)
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n/an/a 75n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197354
PNG
(US9216962, CFH381-M)
Show SMILES Cc1cnc(s1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C16H20N4O3S2/c1-9-8-18-15(24-9)16-19-12(13(25-16)10-5-6-10)14(22)17-7-3-2-4-11(21)20-23/h8,10,23H,2-7H2,1H3,(H,17,22)(H,20,21)
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n/an/a 75n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197365
PNG
(US9216962, CFH455-C)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nc3CCCCc3s2)cc1
Show InChI InChI=1S/C22H22N4O3S2/c27-19(26-29)14-7-5-12(6-8-14)11-23-20(28)17-18(13-9-10-13)31-22(25-17)21-24-15-3-1-2-4-16(15)30-21/h5-8,13,29H,1-4,9-11H2,(H,23,28)(H,26,27)
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n/an/a 75n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM50020904
PNG
(CHEMBL3287262 | US9216962, CFH417)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1Cc1ccccc1)-c1nccs1
Show InChI InChI=1S/C19H20N4O3S2/c24-15(23-26)8-4-5-9-20-17(25)16-14(12-13-6-2-1-3-7-13)28-19(22-16)18-21-10-11-27-18/h1-3,6-7,10-11,26H,4-5,8-9,12H2,(H,20,25)(H,23,24)
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n/an/a 79n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197365
PNG
(US9216962, CFH455-C)
Show SMILES ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nc3CCCCc3s2)cc1
Show InChI InChI=1S/C22H22N4O3S2/c27-19(26-29)14-7-5-12(6-8-14)11-23-20(28)17-18(13-9-10-13)31-22(25-17)21-24-15-3-1-2-4-16(15)30-21/h5-8,13,29H,1-4,9-11H2,(H,23,28)(H,26,27)
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n/an/a 79n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197341
PNG
(US9216962, CFH396)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C17H24N4O3S2/c1-11(2)10-12-14(20-17(26-12)16-19-8-9-25-16)15(23)18-7-5-3-4-6-13(22)21-24/h8-9,11,24H,3-7,10H2,1-2H3,(H,18,23)(H,21,22)
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n/an/a 86n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197357
PNG
(US9216962, CFH407)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCc2s1
Show InChI InChI=1S/C18H22N4O3S2/c23-13(22-25)6-1-2-9-19-16(24)14-15(10-7-8-10)27-18(21-14)17-20-11-4-3-5-12(11)26-17/h10,25H,1-9H2,(H,19,24)(H,22,23)
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n/an/a 86n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM197351
PNG
(US9216962, CFH409-C)
Show SMILES ONC(=O)CCCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C18H24N4O3S2/c23-13(22-25)6-4-2-1-3-5-9-19-16(24)14-15(12-7-8-12)27-18(21-14)17-20-10-11-26-17/h10-12,25H,1-9H2,(H,19,24)(H,22,23)
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n/an/a 86n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020915
PNG
(CHEMBL3287008 | US9216962, CFH412-S)
Show SMILES CC(C)[C@H](NC(=O)c1csc(n1)-c1cscn1)C(=O)OC\C=C\CCS |r|
Show InChI InChI=1S/C17H21N3O3S3/c1-11(2)14(17(22)23-6-4-3-5-7-24)20-15(21)12-9-26-16(19-12)13-8-25-10-18-13/h3-4,8-11,14,24H,5-7H2,1-2H3,(H,20,21)/b4-3+/t14-/m0/s1
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n/an/a 87n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197392
PNG
(US9216962, CFH398-S)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCNC(=O)CS)-c1nccs1
Show InChI InChI=1S/C16H22N4O2S3/c1-10(2)8-11-13(20-16(25-11)15-19-6-7-24-15)14(22)18-5-3-4-17-12(21)9-23/h6-7,10,23H,3-5,8-9H2,1-2H3,(H,17,21)(H,18,22)
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n/an/a 88n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197353
PNG
(US9216962, CFH381-B)
Show SMILES Cc1csc(n1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C16H20N4O3S2/c1-9-8-24-15(18-9)16-19-12(13(25-16)10-5-6-10)14(22)17-7-3-2-4-11(21)20-23/h8,10,23H,2-7H2,1H3,(H,17,22)(H,20,21)
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n/an/a 92n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM197355
PNG
(US9216962, CFH395-M)
Show SMILES Cc1nc(sc1C)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Show InChI InChI=1S/C17H22N4O3S2/c1-9-10(2)25-16(19-9)17-20-13(14(26-17)11-6-7-11)15(23)18-8-4-3-5-12(22)21-24/h11,24H,3-8H2,1-2H3,(H,18,23)(H,21,22)
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n/an/a 97n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 3


(Homo sapiens (Human))		BDBM50020890
PNG
(CHEMBL3287250 | US9216962, CFH382)
Show SMILES CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
Show InChI InChI=1S/C16H22N4O3S2/c1-10(2)9-11-13(19-16(25-11)15-18-7-8-24-15)14(22)17-6-4-3-5-12(21)20-23/h7-8,10,23H,3-6,9H2,1-2H3,(H,17,22)(H,20,21)
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n/an/a 102n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 6


(Homo sapiens (Human))		BDBM197349
PNG
(US9216962, CFH381-C)
Show SMILES ONC(=O)CCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Show InChI InChI=1S/C16H20N4O3S2/c21-11(20-23)4-2-1-3-7-17-14(22)12-13(10-5-6-10)25-16(19-12)15-18-8-9-24-15/h8-10,23H,1-7H2,(H,17,22)(H,20,21)
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n/an/a 105n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
Histone deacetylase 1


(Homo sapiens (Human))		BDBM50020903
PNG
(CHEMBL3287261 | US9216962, CFH448-P)
Show SMILES ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccc(cc1)[N+]([O-])=O)-c1nccs1
Show InChI InChI=1S/C18H17N5O5S2/c24-13(22-26)3-1-2-8-19-16(25)14-15(11-4-6-12(7-5-11)23(27)28)30-18(21-14)17-20-9-10-29-17/h4-7,9-10,26H,1-3,8H2,(H,19,25)(H,22,24)
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n/an/a 105n/an/an/an/an/an/a



Shanghai Puyi Chemical Co., Ltd.

US Patent


Assay Description
Enzyme activity of HDAC1,3 is determined using the substrate Ac-Lys-Tyr-Lys(Ac)-AMC while the enzyme activity of HDAC6 is assayed using the substrate...

US Patent US9216962 (2015)


BindingDB Entry DOI: 10.7270/Q2QJ7G3F
More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%