Affinity Data by Patent

Patent code US9302981

Found 6 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium-dependent serotonin transporter (Homo sapiens (Human))	BDBM215794 (US9302981, 54b) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	22.8	n/a	140	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM215794 (US9302981, 54b) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	45.2	n/a	56.9	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair
Sodium-dependent serotonin transporter (Homo sapiens (Human))	BDBM215795 (US9302981, 54d) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	67.6	n/a	415	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair
Sodium-dependent noradrenaline transporter (Homo sapiens (Human))	BDBM215794 (US9302981, 54b) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	120	n/a	121	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair
Sodium-dependent noradrenaline transporter (Homo sapiens (Human))	BDBM215795 (US9302981, 54d) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	180	n/a	182	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM215795 (US9302981, 54d) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	294	n/a	370	n/a	n/a	n/a	n/a	n/a	n/a
REVIVA PHARMACEUTICALS, Inc. US Patent					Assay Description The radioligand binding assays were carried out at four different test concentrations and the test concentrations were 1 nM, 10 nM, 0.1 μM, and ...				US Patent US9302981 (2016) BindingDB Entry DOI: 10.7270/Q2WS8S3H
REVIVA PHARMACEUTICALS, Inc. US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%