Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224619 (US9326978, 32) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 410 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224617 (US9326978, 30) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 786 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224618 (US9326978, 31) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224621 (US9326978, 34) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM224617 (US9326978, 30) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM224617 (US9326978, 30) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.42E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM224618 (US9326978, 31) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM224619 (US9326978, 32) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224620 (US9326978, 33 | US9326978, 49) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM224620 (US9326978, 33 | US9326978, 49) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 4.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description Each tube in the competitive binding assay contained 100 μl membrane suspension (20 μg protein), 50 μl [125I]-AB-MECA (0.5 nM), and 50... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM224618 (US9326978, 31) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 5.22E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM224621 (US9326978, 34) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM224620 (US9326978, 33 | US9326978, 49) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM224620 (US9326978, 33 | US9326978, 49) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM224621 (US9326978, 34) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM224619 (US9326978, 32) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
The United States of America, Represented by the Secretary, Dept. of Health and Human Services; Universiteit Leiden US Patent | Assay Description For binding to the human A1AR, [3H]R-PIA (2 nM) was incubated with membranes (40 μg/tube) from CHO cells stably expressing the human A1AR at 25°... | US Patent US9326978 (2016) BindingDB Entry DOI: 10.7270/Q2C24V85 | |||||||||||
More data for this Ligand-Target Pair |